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  Subjects -> PHARMACY AND PHARMACOLOGY (Total: 575 journals)
Showing 1 - 200 of 253 Journals sorted by number of followers
Nature Reviews Drug Discovery     Full-text available via subscription   (Followers: 331)
International Journal of Drug Policy     Hybrid Journal   (Followers: 254)
Journal of Clinical Oncology     Hybrid Journal   (Followers: 242)
Journal of Medicinal Chemistry     Hybrid Journal   (Followers: 158)
Journal of Pharmaceutical Sciences     Hybrid Journal   (Followers: 154)
Drugs     Full-text available via subscription   (Followers: 146)
Advanced Drug Delivery Reviews     Hybrid Journal   (Followers: 98)
Pharmaceutical Research     Hybrid Journal   (Followers: 94)
European Journal of Pharmaceutical Sciences     Hybrid Journal   (Followers: 86)
Drug Safety     Full-text available via subscription   (Followers: 83)
Annals of Pharmacotherapy     Hybrid Journal   (Followers: 56)
Biomaterials     Hybrid Journal   (Followers: 54)
Clinical Pharmacology & Therapeutics     Hybrid Journal   (Followers: 44)
Regulatory Toxicology and Pharmacology     Hybrid Journal   (Followers: 42)
Journal of Controlled Release     Hybrid Journal   (Followers: 38)
Annual Review of Pharmacology and Toxicology     Full-text available via subscription   (Followers: 38)
International Journal of Pharmaceutics     Hybrid Journal   (Followers: 37)
Clinical Therapeutics     Hybrid Journal   (Followers: 34)
European Journal of Pharmaceutics and Biopharmaceutics     Hybrid Journal   (Followers: 34)
Pharmacoepidemiology and Drug Safety     Hybrid Journal   (Followers: 33)
British Journal of Clinical Pharmacology     Hybrid Journal   (Followers: 32)
Journal of Pharmacy and Pharmacology     Full-text available via subscription   (Followers: 31)
Drug Development and Industrial Pharmacy     Hybrid Journal   (Followers: 29)
PharmacoEconomics     Full-text available via subscription   (Followers: 27)
Clinical Pharmacokinetics     Full-text available via subscription   (Followers: 27)
AAPS Journal     Hybrid Journal   (Followers: 26)
Critical Reviews in Toxicology     Hybrid Journal   (Followers: 25)
Journal of Clinical Psychopharmacology     Hybrid Journal   (Followers: 24)
International Journal of Pharmacy Practice     Full-text available via subscription   (Followers: 24)
Toxicology and Applied Pharmacology     Hybrid Journal   (Followers: 24)
Chemical Research in Toxicology     Hybrid Journal   (Followers: 22)
Journal of Pharmacokinetics and Pharmacodynamics     Hybrid Journal   (Followers: 22)
Journal of Pain & Palliative Care Pharmacotherapy     Hybrid Journal   (Followers: 21)
Trends in Pharmacological Sciences     Full-text available via subscription   (Followers: 20)
Journal of Applied Toxicology     Hybrid Journal   (Followers: 19)
Journal of Clinical Pharmacology     Hybrid Journal   (Followers: 19)
Pharmaceutical Development and Technology     Hybrid Journal   (Followers: 19)
American Journal of Cardiovascular Drugs     Hybrid Journal   (Followers: 19)
Clinical Trials     Hybrid Journal   (Followers: 18)
Toxicology     Hybrid Journal   (Followers: 18)
Journal of Pharmaceutical and Biomedical Analysis     Hybrid Journal   (Followers: 18)
Clinical Toxicology     Hybrid Journal   (Followers: 18)
International Journal of Toxicology     Hybrid Journal   (Followers: 17)
Critical Reviews in Clinical Laboratory Sciences     Hybrid Journal   (Followers: 16)
Journal of Clinical Pharmacy and Therapeutics     Hybrid Journal   (Followers: 16)
Journal of Natural Products     Hybrid Journal   (Followers: 16)
Pharmaceutical Statistics     Hybrid Journal   (Followers: 15)
Toxicology Letters     Hybrid Journal   (Followers: 15)
Journal of Pharmacy Practice     Hybrid Journal   (Followers: 15)
Psychopharmacology     Hybrid Journal   (Followers: 15)
Basic & Clinical Pharmacology & Toxicology     Hybrid Journal   (Followers: 14)
Cardiovascular Drugs and Therapy     Hybrid Journal   (Followers: 14)
European Journal of Clinical Pharmacology     Hybrid Journal   (Followers: 14)
Current Medicinal Chemistry     Hybrid Journal   (Followers: 13)
American Journal of Therapeutics     Hybrid Journal   (Followers: 13)
Drug and Chemical Toxicology     Hybrid Journal   (Followers: 13)
Journal of the American Pharmacists Association     Full-text available via subscription   (Followers: 13)
Clinical Research and Regulatory Affairs     Hybrid Journal   (Followers: 12)
Seminars in Hematology     Hybrid Journal   (Followers: 12)
Drug Discovery Today: Technologies     Full-text available via subscription   (Followers: 12)
Current Pharmaceutical Design     Hybrid Journal   (Followers: 12)
Journal of Oncology Pharmacy Practice     Hybrid Journal   (Followers: 12)
Journal of Psychopharmacology     Hybrid Journal   (Followers: 11)
Biopharmaceutics and Drug Disposition     Hybrid Journal   (Followers: 11)
Toxicology in Vitro     Hybrid Journal   (Followers: 11)
Drug Development Research     Hybrid Journal   (Followers: 11)
Drug Metabolism and Disposition     Hybrid Journal   (Followers: 11)
Seminars in Oncology Nursing     Full-text available via subscription   (Followers: 10)
Biochemical Pharmacology     Hybrid Journal   (Followers: 10)
Journal of Separation Science     Hybrid Journal   (Followers: 10)
CNS Drugs     Full-text available via subscription   (Followers: 10)
Current Pharmaceutical Biotechnology     Hybrid Journal   (Followers: 10)
Journal of Medical Marketing     Hybrid Journal   (Followers: 10)
Drugs & Aging     Full-text available via subscription   (Followers: 10)
European Neuropsychopharmacology     Hybrid Journal   (Followers: 9)
Food Additives & Contaminants Part A     Hybrid Journal   (Followers: 9)
Journal of Pharmacology and Experimental Therapeutics     Hybrid Journal   (Followers: 9)
Environmental Toxicology and Pharmacology     Hybrid Journal   (Followers: 9)
Medicinal Chemistry     Hybrid Journal   (Followers: 9)
Biometrical Journal     Hybrid Journal   (Followers: 9)
Drugs & Therapy Perspectives     Full-text available via subscription   (Followers: 9)
Prescriber     Hybrid Journal   (Followers: 9)
ChemMedChem     Hybrid Journal   (Followers: 9)
Current Opinion in Pharmacology     Hybrid Journal   (Followers: 9)
European Journal of Pharmacology     Hybrid Journal   (Followers: 8)
Inhalation Toxicology     Hybrid Journal   (Followers: 8)
Antiviral Research     Hybrid Journal   (Followers: 8)
Drug Metabolism Reviews     Hybrid Journal   (Followers: 8)
Progress in Neuro-Psychopharmacology and Biological Psychiatry     Hybrid Journal   (Followers: 8)
Human & Experimental Toxicology     Hybrid Journal   (Followers: 8)
Drug Delivery     Open Access   (Followers: 8)
BioDrugs     Full-text available via subscription   (Followers: 8)
Frontiers in Drug Design & Discovery     Hybrid Journal   (Followers: 8)
Expert Review of Pharmacoeconomics & Outcomes Research     Full-text available via subscription   (Followers: 8)
Experimental and Clinical Psychopharmacology     Full-text available via subscription   (Followers: 7)
Toxicology Mechanisms and Methods     Hybrid Journal   (Followers: 7)
Journal of Pharmacological and Toxicological Methods     Hybrid Journal   (Followers: 7)
Clinical and Experimental Pharmacology and Physiology     Hybrid Journal   (Followers: 7)
Scandinavian Journal of Clinical and Laboratory Investigation     Hybrid Journal   (Followers: 7)
Epilepsy Research     Hybrid Journal   (Followers: 7)
Clinical Drug Investigation     Full-text available via subscription   (Followers: 7)
Journal of Veterinary Pharmacology and Therapeutics     Hybrid Journal   (Followers: 6)
Toxicology and Industrial Health     Hybrid Journal   (Followers: 6)
Skin Pharmacology and Physiology     Full-text available via subscription   (Followers: 6)
Journal of Cardiovascular Pharmacology     Hybrid Journal   (Followers: 6)
AAPS PharmSciTech     Hybrid Journal   (Followers: 6)
Current Drug Discovery Technologies     Hybrid Journal   (Followers: 6)
Anti-Inflammatory & Anti-Allergy Agents in Medicinal Chemistry     Hybrid Journal   (Followers: 6)
Current Therapeutic Research     Open Access   (Followers: 6)
Expert Review of Cardiovascular Therapy     Full-text available via subscription   (Followers: 6)
Current Drug Delivery     Hybrid Journal   (Followers: 6)
Expert Review of Anti-infective Therapy     Full-text available via subscription   (Followers: 5)
Neuropharmacology     Hybrid Journal   (Followers: 5)
Current Drug Metabolism     Hybrid Journal   (Followers: 5)
Fitoterapia     Hybrid Journal   (Followers: 5)
Expert Review of Molecular Diagnostics     Full-text available via subscription   (Followers: 5)
Anti-Infective Agents     Hybrid Journal   (Followers: 5)
Toxicon     Hybrid Journal   (Followers: 5)
Medicinal Research Reviews     Hybrid Journal   (Followers: 5)
Investigational New Drugs     Hybrid Journal   (Followers: 5)
Current Cancer Therapy Reviews     Hybrid Journal   (Followers: 5)
Reviews of Physiology, Biochemistry and Pharmacology     Hybrid Journal   (Followers: 4)
Planta Medica     Hybrid Journal   (Followers: 4)
Current Vascular Pharmacology     Hybrid Journal   (Followers: 4)
Pharmaceutical Medicine     Full-text available via subscription   (Followers: 4)
Journal of Child and Adolescent Psychopharmacology     Hybrid Journal   (Followers: 4)
CNS Drug Reviews     Open Access   (Followers: 4)
Inpharma Weekly     Full-text available via subscription   (Followers: 4)
Journal of Labelled Compounds and Radiopharmaceuticals     Hybrid Journal   (Followers: 4)
Immunopharmacology and Immunotoxicology     Hybrid Journal   (Followers: 4)
International Journal of Pharmaceutical and Healthcare Marketing     Hybrid Journal   (Followers: 4)
Inflammation Research     Hybrid Journal   (Followers: 4)
Cancer Chemotherapy and Pharmacology     Hybrid Journal   (Followers: 4)
International Journal of Neuropsychopharmacology     Open Access   (Followers: 3)
Pharmacology & Therapeutics     Hybrid Journal   (Followers: 3)
Physiology International     Full-text available via subscription   (Followers: 3)
Cardiovascular Therapeutics     Open Access   (Followers: 3)
ASSAY and Drug Development Technologies     Hybrid Journal   (Followers: 3)
Pharmacopsychiatry     Hybrid Journal   (Followers: 3)
Chemotherapy     Full-text available via subscription   (Followers: 3)
Therapeutic Drug Monitoring     Hybrid Journal   (Followers: 3)
Current Drug Therapy     Hybrid Journal   (Followers: 3)
Research in Social and Administrative Pharmacy     Hybrid Journal   (Followers: 3)
PharmacoEconomics & Outcomes News     Full-text available via subscription   (Followers: 3)
Journal of Aerosol Medicine and Pulmonary Drug Delivery     Hybrid Journal   (Followers: 3)
Journal of Ethnopharmacology     Hybrid Journal   (Followers: 3)
Drug Resistance Updates     Hybrid Journal   (Followers: 3)
Journal of Pain Management & Medicine     Open Access   (Followers: 3)
Journal of Infection and Chemotherapy     Hybrid Journal   (Followers: 3)
Journal of Cardiovascular Pharmacology and Therapeutics     Hybrid Journal   (Followers: 3)
Current Pharmacogenomics and Personalized Medicine     Hybrid Journal   (Followers: 3)
Acta Pharmacologica Sinica     Hybrid Journal   (Followers: 3)
Microbial Drug Resistance     Hybrid Journal   (Followers: 3)
Frontiers in Medicinal Chemistry     Hybrid Journal   (Followers: 3)
Human Psychopharmacology Clinical and Experimental     Hybrid Journal   (Followers: 3)
BMC Pharmacology     Open Access   (Followers: 2)
The Brown University Psychopharmacology Update     Hybrid Journal   (Followers: 2)
International Clinical Psychopharmacology     Hybrid Journal   (Followers: 2)
Canadian Journal of Physiology and Pharmacology     Hybrid Journal   (Followers: 2)
Journal of Drug Targeting     Hybrid Journal   (Followers: 2)
Inflammopharmacology     Hybrid Journal   (Followers: 2)
Journal of Inflammation     Open Access   (Followers: 2)
Fundamental & Clinical Pharmacology     Hybrid Journal   (Followers: 2)
Behavioural Pharmacology     Hybrid Journal   (Followers: 2)
Vascular Pharmacology     Hybrid Journal   (Followers: 2)
Pulmonary Pharmacology & Therapeutics     Hybrid Journal   (Followers: 2)
Biomedicine & Pharmacotherapy     Full-text available via subscription   (Followers: 2)
Clinical Neuropharmacology     Hybrid Journal   (Followers: 2)
Drugs in R & D     Full-text available via subscription   (Followers: 2)
International Immunopharmacology     Hybrid Journal   (Followers: 2)
Pharmacology Biochemistry and Behavior     Hybrid Journal   (Followers: 2)
Letters in Drug Design & Discovery     Hybrid Journal   (Followers: 2)
Archiv der Pharmazie     Hybrid Journal   (Followers: 2)
Pharmacological Reviews     Hybrid Journal   (Followers: 2)
Molecular Pharmacology     Hybrid Journal   (Followers: 2)
Journal of Microencapsulation: Microcapsules, Liposomes, Nanoparticles, Microcells, Microspheres     Hybrid Journal   (Followers: 2)
Toxicological & Environmental Chemistry     Hybrid Journal   (Followers: 2)
Particulate Science and Technology: An International Journal     Hybrid Journal   (Followers: 1)
Pharmacological Research     Hybrid Journal   (Followers: 1)
Current Enzyme Inhibition     Hybrid Journal   (Followers: 1)
Journal of Neuroimmune Pharmacology     Hybrid Journal   (Followers: 1)
Current Pharmaceutical Analysis     Hybrid Journal   (Followers: 1)
Current Neuropharmacology     Hybrid Journal   (Followers: 1)
Pharmacogenetics and Genomics     Hybrid Journal   (Followers: 1)
Journal of Texture Studies     Hybrid Journal   (Followers: 1)
Pharmaceutical Biology     Open Access  
Journal of Liposome Research     Hybrid Journal  
Toxin Reviews     Hybrid Journal  
Kaohsiung Journal of Medical Sciences     Open Access  
Redox Report     Open Access  
Pharmacology     Full-text available via subscription  
Pharmaceutical Chemistry Journal     Hybrid Journal  
NeuroMolecular Medicine     Hybrid Journal  
Journal of Ocular Pharmacology and Therapeutics     Hybrid Journal  
Harm Reduction Journal     Open Access  
Current Nanoscience     Hybrid Journal  
Infectious Disorders - Drug Targets     Hybrid Journal  
Current Bioactive Compounds     Hybrid Journal  
Cancer Biotherapy & Radiopharmaceuticals     Hybrid Journal  
Autonomic & Autacoid Pharmacology     Hybrid Journal  

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Similar Journals
Journal Cover
Journal of Medicinal Chemistry
Journal Prestige (SJR): 2.567
Citation Impact (citeScore): 6
Number of Followers: 158  
 
  Hybrid Journal Hybrid journal (It can contain Open Access articles)
ISSN (Print) 0022-2623 - ISSN (Online) 1520-4804
Published by ACS Homepage  [72 journals]
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           and Degrader of Mutant PI3Kα

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      Authors: Emily J. Hanan; Marie-Gabrielle Braun, Robert A. Heald, Calum MacLeod, Connie Chan, Saundra Clausen, Kyle A. Edgar, Charles Eigenbrot, Richard Elliott, Nicholas Endres, Lori S. Friedman, Emily Gogol, Xiao-Hui Gu, Rebecca Hong Thibodeau, Philip S. Jackson, James R. Kiefer, Jamie D. Knight, Michelle Nannini, Raman Narukulla, Amanda Pace⧫, Jodie Pang, Hans E. Purkey, Laurent Salphati, Deepak Sampath, Stephen Schmidt, Steve Sideris, Kyung Song, Swathi Sujatha-Bhaskar, Mark Ultsch, Heidi Wallweber, Jianfeng Xin, SiewKuen Yeap, Amy Young, Yu Zhong, Steven T. Staben
      Abstract: TOC GraphicJournal of Medicinal Chemistry
      DOI : 10.1021/acs.jmedchem.2c01422
      PubDate: Thu, 01 Dec 2022 05:00:00 GMT
       
  • N‑Benzylpiperidinol+Derivatives+as+Potent+and+Selective+USP7+Inhibitors+with+In+Vivo+Antitumor+Immunity+Activity+against+Colon+Cancer&rft.title=Journal+of+Medicinal+Chemistry&rft.issn=0022-2623&rft.date=2022&rft.volume=&rft.aulast=Li&rft.aufirst=Xing&rft.au=Xing+Li&rft.au=Shanlin+Yang,++Honghan+Zhang,++Xipeng+Liu,++Yuchen+Gao,++Yuqi+Chen,++Liu+Liu,++Dalin+Wang,++Zijiang+Liang,++Shengjie+Liu,++Liang+Dai,++Qinglong+Xu,++Haoliang+Yuan,++Caiping+Chen,++Hongbin+Sun,++Xiaoan+Wen">[ASAP] Discovery of Orally Bioavailable N‑Benzylpiperidinol Derivatives
           as Potent and Selective USP7 Inhibitors with In Vivo Antitumor Immunity
           Activity against Colon Cancer

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      Authors: Xing Li; Shanlin Yang, Honghan Zhang, Xipeng Liu, Yuchen Gao, Yuqi Chen, Liu Liu, Dalin Wang, Zijiang Liang, Shengjie Liu, Liang Dai, Qinglong Xu, Haoliang Yuan, Caiping Chen, Hongbin Sun, Xiaoan Wen
      Abstract: TOC GraphicJournal of Medicinal Chemistry
      DOI : 10.1021/acs.jmedchem.2c01444
      PubDate: Thu, 01 Dec 2022 05:00:00 GMT
       
  • [ASAP] Optimization of 1,2,4-Triazole-3-thiones toward Broad-Spectrum
           Metallo-β-lactamase Inhibitors Showing Potent Synergistic Activity on
           VIM- and NDM-1-Producing Clinical Isolates

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      Authors: Alice Legru; Federica Verdirosa, Yen Vo-Hoang, Giusy Tassone, Filippo Vascon, Caitlyn A. Thomas, Filomena Sannio, Giuseppina Corsica, Manuela Benvenuti, Georges Feller, Rémi Coulon, Francesca Marcoccia, Savannah Rowane Devente, Ezeddine Bouajila, Catherine Piveteau, Florence Leroux, Rebecca Deprez-Poulain, Benoît Deprez, Patricia Licznar-Fajardo, Michael W. Crowder, Laura Cendron, Cecilia Pozzi, Stefano Mangani, Jean-Denis Docquier, Jean-François Hernandez, Laurent Gavara
      Abstract: TOC GraphicJournal of Medicinal Chemistry
      DOI : 10.1021/acs.jmedchem.2c01257
      PubDate: Wed, 30 Nov 2022 05:00:00 GMT
       
  • [ASAP] Design and Synthesis of Fibroblast Growth Factor Receptor (FGFR)
           and Histone Deacetylase (HDAC) Dual Inhibitors for the Treatment of Cancer
           

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      Authors: Guoquan Wan; Zhanzhan Feng, Qiangsheng Zhang, Xiao Li, Kai Ran, Huan Feng, Tianwen Luo, Shuyan Zhou, Chang Su, Wei Wei, Ningyu Wang, Chao Gao, Lifeng Zhao, Luoting Yu
      Abstract: TOC GraphicJournal of Medicinal Chemistry
      DOI : 10.1021/acs.jmedchem.2c01413
      PubDate: Wed, 30 Nov 2022 05:00:00 GMT
       
  • [ASAP] Transcriptional Inhibition of MicroRNA miR-122 by Small Molecules
           Reduces Hepatitis C Virus Replication in Liver Cells

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      Authors: Cole Emanuelson; Nicholas Ankenbruck, Rohan Kumbhare, Meryl Thomas, Colleen Connelly, Yasmine Baktash, Glenn Randall, Alexander Deiters
      Abstract: TOC GraphicJournal of Medicinal Chemistry
      DOI : 10.1021/acs.jmedchem.2c01141
      PubDate: Wed, 30 Nov 2022 05:00:00 GMT
       
  • [ASAP] Discovery and Optimization of Potent and Orally Available CTP
           Synthetase Inhibitors for Use in Treatment of Diseases Driven by Aberrant
           Immune Cell Proliferation

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      Authors: Andrew Novak; David Laughton, Rebecca Lane, Emma Blackham, Jennifer Thomas, Elli Chatzopoulou, Joseph Wrigglesworth, Abdul Quddus, Saleh Ahmed, David Cousin, Lorna Duffy, Nathalie Dubois, John Unitt, Katalin Orban, Edward Browne, Michelle Ward, David Mycock, Maria Ieva, Nicholas Bland, Pascal George, Timothy Bourne, Hélène Asnagli, Louise Birch, Geraint Jones
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      DOI : 10.1021/acs.jmedchem.2c01446
      PubDate: Wed, 30 Nov 2022 05:00:00 GMT
       
  • [ASAP] Development of Alkylated Hydrazides as Highly Potent and Selective
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      Abstract: TOC GraphicJournal of Medicinal Chemistry
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  • [ASAP] Recent Update on the Development of PCSK9 Inhibitors for
           Hypercholesterolemia Treatment

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      Authors: Shakir Ahamad; Shahnawaz A. Bhat
      Abstract: TOC GraphicJournal of Medicinal Chemistry
      DOI : 10.1021/acs.jmedchem.2c01290
      PubDate: Tue, 29 Nov 2022 05:00:00 GMT
       
  • N‑Nitrosamines+Derived+from+Active+Pharmaceutical+Ingredients&rft.title=Journal+of+Medicinal+Chemistry&rft.issn=0022-2623&rft.date=2022&rft.volume=&rft.aulast=Ponting&rft.aufirst=David&rft.au=David+J.+Ponting&rft.au=Krista+L.+Dobo¥,++Michelle+O.+Kenyon¥,++Amit+S.+Kalgutkar">[ASAP] Strategies for Assessing Acceptable Intakes for Novel
           N‑Nitrosamines Derived from Active Pharmaceutical Ingredients

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      Authors: David J. Ponting; Krista L. Dobo¥, Michelle O. Kenyon¥, Amit S. Kalgutkar
      Abstract: TOC GraphicJournal of Medicinal Chemistry
      DOI : 10.1021/acs.jmedchem.2c01498
      PubDate: Mon, 28 Nov 2022 05:00:00 GMT
       
  • [ASAP] B‑cell Lymphoma 6 Inhibitors: Current Advances and Prospects of
           Drug Development for Diffuse Large B‑cell Lymphomas

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      Authors: Haijun Gu; Jia He, Yuzhan Li, Dazhao Mi, Tian Guan, Weikai Guo, Bo Liu, Yihua Chen
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      DOI : 10.1021/acs.jmedchem.2c01433
      PubDate: Mon, 28 Nov 2022 05:00:00 GMT
       
  • In+Vivo+Evaluation+of+Novel+C‑17+Amine+Derivatives+Based+on+GSK3640254+as+HIV‑1+Maturation+Inhibitors+with+Broad+Spectrum+Activity&rft.title=Journal+of+Medicinal+Chemistry&rft.issn=0022-2623&rft.date=2022&rft.volume=&rft.aulast=Hartz&rft.aufirst=Richard&rft.au=Richard+A.+Hartz&rft.au=Li+Xu,++Sing-Yuen+Sit,++Jie+Chen,++Brian+L.+Venables,++Zeyu+Lin,++Sharon+Zhang,++Zhufang+Li,++Dawn+Parker,++Tara+S.+Simmons,++Susan+Jenkins,++Umesh+M.+Hanumegowda,++Ira+Dicker,++Mark+Krystal,++Nicholas+A.+Meanwell,++Alicia+Regueiro-Ren">[ASAP] Synthesis, Structure–Activity Relationships, and In Vivo
           Evaluation of Novel C‑17 Amine Derivatives Based on GSK3640254 as
           HIV‑1 Maturation Inhibitors with Broad Spectrum Activity

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      Authors: Richard A. Hartz; Li Xu, Sing-Yuen Sit, Jie Chen, Brian L. Venables, Zeyu Lin, Sharon Zhang, Zhufang Li, Dawn Parker, Tara S. Simmons, Susan Jenkins, Umesh M. Hanumegowda, Ira Dicker, Mark Krystal, Nicholas A. Meanwell, Alicia Regueiro-Ren
      Abstract: TOC GraphicJournal of Medicinal Chemistry
      DOI : 10.1021/acs.jmedchem.2c01618
      PubDate: Mon, 28 Nov 2022 05:00:00 GMT
       
  • [ASAP] Making Protein Degradation Visible: Discovery of Theranostic
           PROTACs for Detecting and Degrading NAMPT

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      Authors: Junfei Cheng; Shipeng He, Jun Xu, Min Huang, Guoqiang Dong, Chunquan Sheng
      Abstract: TOC GraphicJournal of Medicinal Chemistry
      DOI : 10.1021/acs.jmedchem.2c01243
      PubDate: Mon, 28 Nov 2022 05:00:00 GMT
       
  • [ASAP] What We Have Gained from Ibogaine: α3β4 Nicotinic Acetylcholine
           Receptor Inhibitors as Treatments for Substance Use Disorders

    • Free pre-print version: Loading...

      Authors: Carolyn J. Straub; Lisa E. Rusali, Kyle M. Kremiller, Andrew P. Riley
      Abstract: TOC GraphicJournal of Medicinal Chemistry
      DOI : 10.1021/acs.jmedchem.2c01562
      PubDate: Mon, 28 Nov 2022 05:00:00 GMT
       
  • [ASAP] Membrane-Active Cyclic Amphiphilic Peptides: Broad-Spectrum
           Antibacterial Activity Alone and in Combination with Antibiotics

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      Authors: Eman H. M. Mohammed; Sandeep Lohan, Tarra Ghaffari, Shilpi Gupta, Rakesh K. Tiwari, Keykavous Parang
      Abstract: TOC GraphicJournal of Medicinal Chemistry
      DOI : 10.1021/acs.jmedchem.2c01469
      PubDate: Mon, 28 Nov 2022 05:00:00 GMT
       
  • [ASAP] Synthesis and Characterization of NUC-7738, an Aryloxy
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    • Free pre-print version: Loading...

      Authors: Michaela Serpi; Valentina Ferrari, Christopher McGuigan, Essam Ghazaly, Chris Pepper
      Abstract: TOC GraphicJournal of Medicinal Chemistry
      DOI : 10.1021/acs.jmedchem.2c01348
      PubDate: Wed, 23 Nov 2022 05:00:00 GMT
       
  • [ASAP] Correction to “Rational Design, Synthesis, and Biological
           Evaluation of Novel S1PR2 Antagonists for Reversing 5‑FU-Resistance in
           Colorectal Cancer”

    • Free pre-print version: Loading...

      Authors: Dongdong Luo; Xiaochun Liu, Leilei Jiang, Zhikun Guo, Yan Lv, Xiaochen Tian, Xiaoyan Wang, Shuxiang Cui, Shengbiao Wan, Ximing Xu, Xiaoyang Li, Xianjun Qu
      Abstract: Journal of Medicinal Chemistry
      DOI : 10.1021/acs.jmedchem.2c01832
      PubDate: Wed, 23 Nov 2022 05:00:00 GMT
       
  • [ASAP] Development and Utility of a PAK1-Selective Degrader

    • Free pre-print version: Loading...

      Authors: Hoi-Yee Chow; Sofiia Karchugina, Brian J. Groendyke, Sean Toenjes, John Hatcher, Katherine A. Donovan, Eric S. Fischer, Gleb Abalakov, Bulat Faezov, Roland Dunbrack, Nathanael S. Gray, Jonathan Chernoff
      Abstract: TOC GraphicJournal of Medicinal Chemistry
      DOI : 10.1021/acs.jmedchem.2c00756
      PubDate: Wed, 23 Nov 2022 05:00:00 GMT
       
  • [ASAP] Identification of a Novel Potent CYP4Z1 Inhibitor Attenuating the
           Stemness of Breast Cancer Cells through Lead Optimization

    • Free pre-print version: Loading...

      Authors: Yin Yuan; Hong Yao, Manzhen Zhou, Xiaoqian Ma, Yi Zhou, Jinyi Xu, Miaomiao Niu, Jun Yin, Lufeng Zheng, Shengtao Xu
      Abstract: TOC GraphicJournal of Medicinal Chemistry
      DOI : 10.1021/acs.jmedchem.2c01320
      PubDate: Tue, 22 Nov 2022 05:00:00 GMT
       
  • [ASAP] Riboflavin-Promoted In Situ Photoactivation of Dihydroalkaloid
           Prodrugs for Cancer Therapy

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      Authors: Xin Yang; Limin Ma, Hongwei Shao, Zikai Zhou, Xia Ling, Mengyu Yao, Guowen Luo, Stefano Scoditti, Emilia Sicilia, Gloria Mazzone, Meng Gao, Ben Zhong Tang
      Abstract: TOC GraphicJournal of Medicinal Chemistry
      DOI : 10.1021/acs.jmedchem.2c01262
      PubDate: Mon, 21 Nov 2022 05:00:00 GMT
       
  • [ASAP] Identification and Characterization of a Novel Indoleamine
           2,3-Dioxygenase 1 Protein Degrader for Glioblastoma

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      Authors: Lakshmi R. Bollu; Prashant V. Bommi, Paige J. Monsen, Lijie Zhai, Kristen L. Lauing, April Bell, Miri Kim, Erik Ladomersky, Xinyu Yang, Leonidas C. Platanias, Daniela E. Matei, Marcelo G. Bonini, Hidayatullah G. Munshi, Rintaro Hashizume, Jennifer D. Wu⧫, Bin Zhang⧫, Charles David James, Peiwen Chen, Masha Kocherginsky, Craig Horbinski, Michael D. Cameron, Arabela A. Grigorescu, Bakhtiar Yamini, Rimas V. Lukas, Gary E. Schiltz, Derek A. Wainwright⧫
      Abstract: TOC GraphicJournal of Medicinal Chemistry
      DOI : 10.1021/acs.jmedchem.2c00771
      PubDate: Mon, 21 Nov 2022 05:00:00 GMT
       
  • [ASAP] Lead Optimization and Avoidance of Metabolic-perturbing Motif
           Developing Novel Diarylpyrimidines as Potent HIV‑1 NNRTIs

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      Authors: Yanying Sun; Zhenzhen Zhou, Da Feng, Lanlan Jing, Fabao Zhao, Zhao Wang, Tao Zhang, Hao Lin, Hao Song, Erik De Clercq, Christophe Pannecouque, Peng Zhan, Xinyong Liu, Dongwei Kang
      Abstract: TOC GraphicJournal of Medicinal Chemistry
      DOI : 10.1021/acs.jmedchem.2c00576
      PubDate: Mon, 21 Nov 2022 05:00:00 GMT
       
  • [ASAP] JDQ443, a Structurally Novel, Pyrazole-Based, Covalent Inhibitor of
           KRASG12C for the Treatment of Solid Tumors

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      Authors: Edwige Lorthiois; Marc Gerspacher, Kim S. Beyer, Andrea Vaupel, Catherine Leblanc, Rowan Stringer, Andreas Weiss, Rainer Wilcken, Daniel A. Guthy, Andreas Lingel, Claudio Bomio-Confaglia, Rainer Machauer, Pascal Rigollier, Johannes Ottl, Dorothee Arz, Pascal Bernet, Gaëlle Desjonqueres, Solene Dussauge, Malika Kazic-Legueux, Marie-Anne Lozac’h, Christophe Mura, Mickaël Sorge, Milen Todorov, Nicolas Warin, Florence Zink, Hans Voshol, Frederic J. Zecri, Richard C. Sedrani, Nils Ostermann, Saskia M. Brachmann, Simona Cotesta
      Abstract: TOC GraphicJournal of Medicinal Chemistry
      DOI : 10.1021/acs.jmedchem.2c01438
      PubDate: Fri, 18 Nov 2022 05:00:00 GMT
       
  • N‑Acyl-6-sulfonamide-tetrahydroquinoline+Derivatives+as+Novel+Non-Steroidal+Selective+Glucocorticoid+Receptor+Modulators&rft.title=Journal+of+Medicinal+Chemistry&rft.issn=0022-2623&rft.date=2022&rft.volume=&rft.aulast=Li&rft.aufirst=Dan&rft.au=Dan+Li&rft.au=Xiaodong+Bao,++Jinping+Pang,++Xueping+Hu,++Longling+Wang,++Jiajia+Wang,++Zhaoxu+Yang,++Lei+Xu,++Siyu+Wang,++Qinjie+Weng,++Sunliang+Cui,++Tingjun+Hou">[ASAP] Discovery and Optimization of
           N‑Acyl-6-sulfonamide-tetrahydroquinoline Derivatives as Novel
           Non-Steroidal Selective Glucocorticoid Receptor Modulators

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      Authors: Dan Li; Xiaodong Bao, Jinping Pang, Xueping Hu, Longling Wang, Jiajia Wang, Zhaoxu Yang, Lei Xu, Siyu Wang, Qinjie Weng, Sunliang Cui, Tingjun Hou
      Abstract: TOC GraphicJournal of Medicinal Chemistry
      DOI : 10.1021/acs.jmedchem.2c01082
      PubDate: Fri, 18 Nov 2022 05:00:00 GMT
       
  • [ASAP] Synthesis and Evaluation of Polymyxins Bearing Reductively Labile
           Disulfide-Linked Lipids

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      Authors: Cornelis J. Slingerland; Charlotte M. J. Wesseling, Paolo Innocenti, Koen G. C. Westphal, Rosalinde Masereeuw, Nathaniel I. Martin
      Abstract: TOC GraphicJournal of Medicinal Chemistry
      DOI : 10.1021/acs.jmedchem.2c01528
      PubDate: Fri, 18 Nov 2022 05:00:00 GMT
       
  • N‑(5-(Pyridin-3-yl)‑1H‑indazol-3-yl)benzamide+Derivatives+as+Potent+Cyclin-Dependent+Kinase+7+Inhibitors+for+the+Treatment+of+Autosomal+Dominant+Polycystic+Kidney+Disease&rft.title=Journal+of+Medicinal+Chemistry&rft.issn=0022-2623&rft.date=2022&rft.volume=&rft.aulast=Yang&rft.aufirst=Bowen&rft.au=Bowen+Yang&rft.au=Haoran+Zhang,++Na+Li,++Lixin+Gao,++Hong+Jiang,++Weijuan+Kan,++Haoxing+Yuan,++Jia+Li,++Dongmei+Zhao,++Bing+Xiong,++Yubo+Zhou,++Dong+Guo,++Tongchao+Liu">[ASAP] Discovery of Novel
           N‑(5-(Pyridin-3-yl)‑1H‑indazol-3-yl)benzamide Derivatives as Potent
           Cyclin-Dependent Kinase 7 Inhibitors for the Treatment of Autosomal
           Dominant Polycystic Kidney Disease

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      Authors: Bowen Yang; Haoran Zhang, Na Li, Lixin Gao, Hong Jiang, Weijuan Kan, Haoxing Yuan, Jia Li, Dongmei Zhao, Bing Xiong, Yubo Zhou, Dong Guo, Tongchao Liu
      Abstract: TOC GraphicJournal of Medicinal Chemistry
      DOI : 10.1021/acs.jmedchem.2c01334
      PubDate: Thu, 17 Nov 2022 05:00:00 GMT
       
  • H‑pyrazole-3-carboxyl+Derivatives+as+Potent+P2Y14R+Antagonists+with+Anti-Inflammatory+Characters&rft.title=Journal+of+Medicinal+Chemistry&rft.issn=0022-2623&rft.date=2022&rft.volume=&rft.aulast=Wang&rft.aufirst=Yu-hang&rft.au=Yu-hang+Wang&rft.au=Meng-ze+Zhou,++Tao+Ye,++Ping-ping+Wang,++Ran+Lu,++Yi-lin+Wang,++Chun-xiao+Liu,++Wen+Xiao,++Jia-yi+Li,++Zi-bo+Meng,++Li-li+Xu,++Qing-hua+Hu,++Cheng+Jiang">[ASAP] Discovery of a Series of 5‑Amide‑1H‑pyrazole-3-carboxyl
           Derivatives as Potent P2Y14R Antagonists with Anti-Inflammatory Characters
           

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      Authors: Yu-hang Wang; Meng-ze Zhou, Tao Ye, Ping-ping Wang, Ran Lu, Yi-lin Wang, Chun-xiao Liu, Wen Xiao, Jia-yi Li, Zi-bo Meng, Li-li Xu, Qing-hua Hu, Cheng Jiang
      Abstract: TOC GraphicJournal of Medicinal Chemistry
      DOI : 10.1021/acs.jmedchem.2c01632
      PubDate: Thu, 17 Nov 2022 05:00:00 GMT
       
  • [ASAP] Induction of Ferroptosis in Glioblastoma and Ovarian Cancers by a
           New Pyrrole Tubulin Assembly Inhibitor

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      Authors: Michela Puxeddu; Jianchao Wu, Ruoli Bai, Michele D’Ambrosio, Marianna Nalli, Antonio Coluccia, Simone Manetto, Alessia Ciogli, Domiziana Masci, Andrea Urbani, Cinzia Fionda, Sonia Coni, Rosa Bordone, Gianluca Canettieri, Chiara Bigogno, Giulio Dondio, Ernest Hamel, Te Liu, Romano Silvestri, Giuseppe La Regina
      Abstract: TOC GraphicJournal of Medicinal Chemistry
      DOI : 10.1021/acs.jmedchem.2c01457
      PubDate: Thu, 17 Nov 2022 05:00:00 GMT
       
  • [ASAP] Discovery of ABBV-3373, an Anti-TNF Glucocorticoid Receptor
           Modulator Immunology Antibody Drug Conjugate

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      Authors: Adrian D. Hobson; Michael J. McPherson, Martin E. Hayes, Christian Goess, Xiang Li, Jian Zhou, Zhongyuan Wang, Yajie Yu, Jindong Yang, Liang Sun, Qiang Zhang, Pei Qu, Shi Yang, Axel Hernandez, Jr., Shaughn H. Bryant, Suzanne L. Mathieu, Agnieszka K. Bischoff, Julia Fitzgibbons, Ling C. Santora, Lu Wang, Lu Wang, Margaret M. Fettis, Xiaofeng Li, Christopher C. Marvin, Zhi Wang, Meena V. Patel, Diana L. Schmidt, Tongmei Li, John T. Randolph, Rodger F. Henry, Candace Graff, Yu Tian, Ana L. Aguirre, Anurupa Shrestha
      Abstract: TOC GraphicJournal of Medicinal Chemistry
      DOI : 10.1021/acs.jmedchem.2c01579
      PubDate: Thu, 17 Nov 2022 05:00:00 GMT
       
  • [ASAP] Design and Structural Optimization of Orally Bioavailable SOS1
           Inhibitors for the Treatment of KRAS-Driven Carcinoma

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      Authors: Silong Zhang; Yu Zhang, Xin Chen, Juan Xu, Huaxiang Fang, Yuanyuan Li, Yi Liu, Huan He
      Abstract: TOC GraphicJournal of Medicinal Chemistry
      DOI : 10.1021/acs.jmedchem.2c01517
      PubDate: Thu, 17 Nov 2022 05:00:00 GMT
       
  • [ASAP] Targeting Gatekeeper Mutations for Kinase Drug Discovery

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      Authors: Yang Zhou; Shuang Xiang, Fang Yang, Xiaoyun Lu
      Abstract: TOC GraphicJournal of Medicinal Chemistry
      DOI : 10.1021/acs.jmedchem.2c01361
      PubDate: Thu, 17 Nov 2022 05:00:00 GMT
       
  • [ASAP] Structure-Guided Design of Halofuginone Derivatives as ATP-Aided
           Inhibitors Against Bacterial Prolyl-tRNA Synthetase

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      Authors: Bao Cheng; Zhengjun Cai, Ziqing Luo, Siting Luo, Zhiteng Luo, Yanfang Cheng, Ying Yu, Junsong Guo, Yingchen Ju, Qiong Gu, Jun Xu, Xianxing Jiang, Geng Li, Huihao Zhou
      Abstract: TOC GraphicJournal of Medicinal Chemistry
      DOI : 10.1021/acs.jmedchem.2c01496
      PubDate: Thu, 17 Nov 2022 05:00:00 GMT
       
  • [ASAP] Engineering the Cyclization Loop of MCoTI-II Generates Targeted
           Cyclotides that Potently Inhibit Factor XIIa

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      Authors: Sixin Tian; Thomas Durek, Conan K. Wang, Christina N. Zdenek, Bryan G. Fry, David J. Craik, Simon J. de Veer
      Abstract: TOC GraphicJournal of Medicinal Chemistry
      DOI : 10.1021/acs.jmedchem.2c01080
      PubDate: Wed, 16 Nov 2022 05:00:00 GMT
       
  • [ASAP] Macrocyclization of Quinazoline-Based EGFR Inhibitors Leads to
           Exclusive Mutant Selectivity for EGFR L858R and Del19

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      Authors: Jennifer A. Amrhein; Tyler S. Beyett, William W. Feng, Andreas Krämer, Janik Weckesser, Ilse K. Schaeffner, Jaimin K. Rana, Pasi A. Jänne, Michael J. Eck, Stefan Knapp, Thomas Hanke
      Abstract: TOC GraphicJournal of Medicinal Chemistry
      DOI : 10.1021/acs.jmedchem.2c01041
      PubDate: Wed, 16 Nov 2022 05:00:00 GMT
       
  • Pseudomonas+aeruginosa+and+Methicillin-Resistant+Staphylococcus+aureus+Infections&rft.title=Journal+of+Medicinal+Chemistry&rft.issn=0022-2623&rft.date=2022&rft.volume=&rft.aulast=Guo&rft.aufirst=Xiaomin&rft.au=Xiaomin+Guo&rft.au=Tiantian+Yan,++Jing+Rao,++Yingying+An,++Xin+Yue,++Xiaokang+Miao,++Rui+Wang,++Wangsheng+Sun,++Jianfeng+Cai,++Junqiu+Xie">[ASAP] Novel Feleucin-K3-Derived Peptides Modified with Sulfono-γ-AA
           Building Blocks Targeting Pseudomonas aeruginosa and Methicillin-Resistant
           Staphylococcus aureus Infections

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      Authors: Xiaomin Guo; Tiantian Yan, Jing Rao, Yingying An, Xin Yue, Xiaokang Miao, Rui Wang, Wangsheng Sun, Jianfeng Cai, Junqiu Xie
      Abstract: TOC GraphicJournal of Medicinal Chemistry
      DOI : 10.1021/acs.jmedchem.2c01396
      PubDate: Wed, 09 Nov 2022 05:00:00 GMT
       
  • [ASAP] Imaging Leucine-Rich Repeat Kinase 2 In Vivo with 18F‑Labeled
           Positron Emission Tomography Ligand

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      Authors: Zhen Chen; Jiahui Chen, Laigao Chen, Chi-Hyeon Yoo, Jian Rong, Hualong Fu, Tuo Shao, Karen Coffman, Stefanus J. Steyn, April T. Davenport, James B. Daunais, Ahmed Haider, Lee Collier, Lee Josephson, Hsiao-Ying Wey, Lei Zhang, Steven H. Liang
      Abstract: TOC GraphicJournal of Medicinal Chemistry
      DOI : 10.1021/acs.jmedchem.2c00551
      PubDate: Tue, 18 Oct 2022 04:00:00 GMT
       
  • [ASAP] Mechanism of Action and Structure–Activity Relationship of
           α‑Conotoxin Mr1.1 at the Human α9α10 Nicotinic Acetylcholine Receptor
           

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      Authors: Jiazhen Liang; Han-Shen Tae, Zitong Zhao, Xiao Li, Jinghui Zhang, Shen Chen, Tao Jiang, David J. Adams, Rilei Yu
      Abstract: TOC GraphicJournal of Medicinal Chemistry
      DOI : 10.1021/acs.jmedchem.2c00494
      PubDate: Thu, 22 Sep 2022 04:00:00 GMT
       
  • [ASAP] Magnet for the Needle in Haystack: “Crystal Structure First”
           Fragment Hits Unlock Active Chemical Matter Using Targeted Exploration of
           Vast Chemical Spaces

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      Authors: Janis Müller; Raphael Klein, Olga Tarkhanova, Anastasiia Gryniukova, Petro Borysko, Stefan Merkl, Moritz Ruf, Alexander Neumann, Marcus Gastreich, Yurii S. Moroz, Gerhard Klebe, Serghei Glinca
      Abstract: TOC GraphicJournal of Medicinal Chemistry
      DOI : 10.1021/acs.jmedchem.2c00813
      PubDate: Wed, 07 Sep 2022 04:00:00 GMT
       
  • [ASAP] Non-Covalent Albumin Ligands in FDA-Approved Therapeutic Peptides
           and Proteins

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      Authors: Florencio Zaragoza
      Abstract: TOC GraphicJournal of Medicinal Chemistry
      DOI : 10.1021/acs.jmedchem.2c01021
      PubDate: Fri, 12 Aug 2022 04:00:00 GMT
       
 
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