Subjects -> CHEMISTRY (Total: 986 journals)
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    - ORGANIC CHEMISTRY (47 journals)
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ORGANIC CHEMISTRY (47 journals)

Showing 1 - 41 of 41 Journals sorted alphabetically
ACS Omega     Open Access   (Followers: 2)
Advances in Image and Video Processing     Open Access   (Followers: 18)
Advances in Physical Organic Chemistry     Full-text available via subscription   (Followers: 4)
Advances in Redox Research     Open Access   (Followers: 4)
American Journal of Organic Chemistry     Open Access   (Followers: 15)
Asian Journal of Organic Chemistry     Hybrid Journal   (Followers: 4)
Beilstein Journal of Organic Chemistry     Open Access   (Followers: 13)
Biochemia Medica     Open Access  
Current Organic Chemistry     Hybrid Journal   (Followers: 14)
Current Organic Synthesis     Hybrid Journal   (Followers: 12)
European Journal of Organic Chemistry     Hybrid Journal   (Followers: 59)
Herbal Medicine: Open Access     Open Access  
International Journal of Organic Chemistry     Open Access   (Followers: 9)
International Journal of Polymeric Materials     Hybrid Journal   (Followers: 6)
Journal of Bioactive and Compatible Polymers     Hybrid Journal   (Followers: 2)
Journal of Biomaterials Science, Polymer Edition     Hybrid Journal   (Followers: 9)
Journal of Organic Semiconductors     Open Access   (Followers: 6)
Journal of Peptide Science     Hybrid Journal   (Followers: 14)
Journal of Physical Organic Chemistry     Hybrid Journal   (Followers: 8)
Journal of Physiology and Biochemistry     Hybrid Journal   (Followers: 3)
Journal of Progressive Research in Chemistry     Open Access  
Journal of Proteins and Proteomics     Open Access   (Followers: 2)
Mini-Reviews in Organic Chemistry     Hybrid Journal   (Followers: 10)
Nigerian Journal of Chemical Research     Full-text available via subscription   (Followers: 1)
Open Journal of Organic Polymer Materials     Open Access   (Followers: 1)
Organic & Biomolecular Chemistry     Hybrid Journal   (Followers: 56)
Organic and Medicinal Chemistry Letters     Open Access   (Followers: 5)
Organic Chemistry : Current Research     Open Access   (Followers: 12)
Organic Chemistry Frontiers     Hybrid Journal   (Followers: 9)
Organic Chemistry International     Open Access   (Followers: 7)
Organic Geochemistry     Hybrid Journal   (Followers: 3)
Organic Letters     Hybrid Journal   (Followers: 92)
Organic Preparations and Procedures International: The New Journal for Organic Synthesis     Hybrid Journal   (Followers: 3)
Organic Process Research & Development     Hybrid Journal   (Followers: 32)
Progress in Organic Coatings     Hybrid Journal   (Followers: 7)
Reports in Organic Chemistry     Open Access   (Followers: 7)
Russian Journal of Organic Chemistry     Hybrid Journal   (Followers: 3)
Synthetic Communications: An International Journal for Rapid Communication of Synthetic Organic Chemistry     Hybrid Journal   (Followers: 31)
The Journal of Organic Chemistry     Hybrid Journal   (Followers: 135)
Vibrational Spectroscopy     Hybrid Journal   (Followers: 11)
World Journal of Organic Chemistry     Open Access   (Followers: 5)
Similar Journals
Journal Cover
Organic Process Research & Development
Journal Prestige (SJR): 1.405
Citation Impact (citeScore): 3
Number of Followers: 32  
 
  Hybrid Journal Hybrid journal (It can contain Open Access articles)
ISSN (Print) 1083-6160 - ISSN (Online) 1520-586X
Published by ACS Homepage  [68 journals]
  • [ASAP] When Safety Data Sheets are a Safety Hazard

    • Free pre-print version: Loading...

      Authors: Alexander G. Kolchinski
      Abstract: TOC GraphicOrganic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00427
      PubDate: Fri, 14 Jan 2022 05:00:00 GMT
       
  • [ASAP] Improved Purification of GalNAc-Conjugated Antisense
           Oligonucleotides Using Boronic Acids

    • Free pre-print version: Loading...

      Authors: Christopher M. Gabriel; Brian R. Pimentel, Christian A. Gomez, Isaiah Cedillo, Andrew A. Rodriguez
      Abstract: TOC GraphicOrganic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00439
      PubDate: Wed, 12 Jan 2022 05:00:00 GMT
       
  • [ASAP] Application of a Statistical Approach to Process Development of
           Futibatinib by Employing Quality-by-Design Principles. Part 3: Development
           of Design Space for Control of Particle Size Distribution

    • Free pre-print version: Loading...

      Authors: Yasunori Abe; Kosuke Emori
      Abstract: TOC GraphicOrganic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00147
      PubDate: Wed, 12 Jan 2022 05:00:00 GMT
       
  • [ASAP] Application of a Statistical Approach to the Process Development of
           Futibatinib by Employing Quality-by-Design Principles. Part 2: Development
           of Design Space for Impurities Using the Response Surface Methodology

    • Free pre-print version: Loading...

      Authors: Yasunori Abe; Kosuke Emori
      Abstract: TOC GraphicOrganic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00146
      PubDate: Wed, 12 Jan 2022 05:00:00 GMT
       
  • [ASAP] Application of a Statistical Approach to Process Development of
           Futibatinib by Employing Quality-by-Design Principles. Part 1:
           Identification of Critical Process Parameters for Impurities

    • Free pre-print version: Loading...

      Authors: Yasunori Abe; Kosuke Emori
      Abstract: TOC GraphicOrganic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00145
      PubDate: Wed, 12 Jan 2022 05:00:00 GMT
       
  • [ASAP] Convenient, Large-Scale Synthesis of (S)TRIP Using Suzuki
           Cross-Coupling Conditions

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      Authors: Ramesh Mamidala; Chandrasekhar Kommuri, Justin Paulose, Hema Aswath, Lokesh Pawar, Athimoolam Arunachalampillai, Alan H. Cherney, Jason S. Tedrow, Andreas R. Rötheli, Adrian Ortiz
      Abstract: TOC GraphicOrganic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00386
      PubDate: Mon, 10 Jan 2022 05:00:00 GMT
       
  • [ASAP] Stirring Peptide Synthesis to a New Level of Efficiency

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      Authors: Johnny N. Naoum; Israel Alshanski, Guy Mayer, Poriah Strauss, Mattan Hurevich
      Abstract: TOC GraphicOrganic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00304
      PubDate: Mon, 10 Jan 2022 05:00:00 GMT
       
  • [ASAP] Facile and Scalable Methodology for the
           Pyrrolo[2,1f][1,2,4]triazine of Remdesivir

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      Authors: Sarabindu Roy; Ajay Yadaw, Subho Roy, Gopal Sirasani, Aravind Gangu, Jack D. Brown, Joseph D. Armstrong, III, Rodger W. Stringham, B. Frank Gupton, Chris H. Senanayake, David R. Snead
      Abstract: TOC GraphicOrganic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00071
      PubDate: Fri, 07 Jan 2022 05:00:00 GMT
       
  • [ASAP] Rapid Continuous-Flow Water-Free Synthesis of Ultrapure Ionic
           Liquids Assisted by Microwaves

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      Authors: Lei Cao; Hong Won Kim, Yu Jin Jeong, Seung Chang Han, Jin Kyoon Park
      Abstract: TOC GraphicOrganic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00412
      PubDate: Fri, 07 Jan 2022 05:00:00 GMT
       
  • [ASAP] Some Items of Interest to Process R&D Chemists and Engineers

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      Authors: Paul F. Richardson; Alan Steven, Robert B. Kargbo, Carlos Mateos, Andrei A. Zlota, Christopher C. Nawrat, Antonio Ramirez, John Knight
      Abstract: Organic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00482
      PubDate: Wed, 05 Jan 2022 05:00:00 GMT
       
  • [ASAP] Scalable and Safe Transformation of 3Hydroxypropionitrile to Its
           Amidoxime

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      Authors: Leah N. Hlubb; Eric C. Johnson, Jesse J. Sabatini, Joshua A. Orlicki
      Abstract: TOC GraphicOrganic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00401
      PubDate: Mon, 03 Jan 2022 05:00:00 GMT
       
  • [ASAP] Quantum Mechanical Methods for Thermal Hazard Risk Assessment in
           Early Phase Pharmaceutical Development

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      Authors: Fareed Bhasha Sayyed; Stanley P. Kolis, Han Xia
      Abstract: TOC GraphicOrganic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00391
      PubDate: Mon, 03 Jan 2022 05:00:00 GMT
       
  • [ASAP] Optimization of the Everolimus Intermediate Preparation Process:
           Impurity Identification Followed by One-Pot Transformation to the Desired
           Product

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      Authors: Aleksandr N. Shestakov; Murat B. Supurgibekov, Elena A. Shpakova, Dmitrii E. Sharkov
      Abstract: TOC GraphicOrganic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00456
      PubDate: Fri, 31 Dec 2021 05:00:00 GMT
       
  • [ASAP] Sulfone Displacement Approach for Large-Scale Synthesis of
           4ChloroN(1-methyl1Hpyrazol-4-yl)pyrimidin-2-amine

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      Authors: Chaomin Li; Fredrik Haeffner, Shujun Wang, Cuicui Yuan, Deju Shang, Xianglin Shi, Bin Ma, Brian T. Hopkins, Erin M. O’Brien
      Abstract: TOC GraphicOrganic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00314
      PubDate: Thu, 30 Dec 2021 05:00:00 GMT
       
  • [ASAP] Tetrahydro4Hpyran-4-one: From the Laboratory Scale to Pilot Plant
           Manufacture

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      Authors: Sara Zahim; Kenny Delacroix, Agathe Carlier, Thierry Berranger, Julie Bergraser, Pierre-Georges Echeverria, Laurent Petit
      Abstract: TOC GraphicOrganic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00403
      PubDate: Wed, 29 Dec 2021 05:00:00 GMT
       
  • [ASAP] Real-Time Monitoring of Continuous Pharmaceutical Mixed Suspension
           Mixed Product Removal Crystallization Using Image Analysis

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      Authors: András Domokos; Lajos Madarász, György Stoffán, Kornélia Tacsi, Dorián Galata, Kristóf Csorba, Panna Vass, Zsombor K. Nagy, Hajnalka Pataki
      Abstract: TOC GraphicOrganic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00372
      PubDate: Wed, 29 Dec 2021 05:00:00 GMT
       
  • [ASAP] Recent Advances in Nonprecious Metal Catalysis

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      Authors: Shashank Shekhar; Tonia S. Ahmed, Andrew R. Ickes, Michael C. Haibach
      Abstract: TOC GraphicOrganic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00410
      PubDate: Wed, 29 Dec 2021 05:00:00 GMT
       
  • N,N-Dimethylformamide&rft.title=Organic+Process+Research+&+Development&rft.issn=1083-6160&rft.date=2021&rft.volume=&rft.aulast=Leko&rft.aufirst=Maria&rft.au=Maria+Leko&rft.au=Polina+Filippova,++Marina+Dorosh,++Karin+Rustler,++Thomas+Bruckdorfer,++Sergey+Burov">[ASAP] 2-Chlorotrityl Chloride and 4-Methylbenzhydryl Bromide Resin
           Loading Using the Mixture of Organic Solvents: A “Greener” Alternative
           to Dichloromethane and N,N-Dimethylformamide

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      Authors: Maria Leko; Polina Filippova, Marina Dorosh, Karin Rustler, Thomas Bruckdorfer, Sergey Burov
      Abstract: TOC GraphicOrganic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00356
      PubDate: Mon, 27 Dec 2021 05:00:00 GMT
       
  • [ASAP] Coprecipitated Amorphous Dispersions as Drug Substance:
           Opportunities and Challenges

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      Authors: Neil A. Strotman; Luke Schenck
      Abstract: TOC GraphicOrganic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00380
      PubDate: Thu, 23 Dec 2021 05:00:00 GMT
       
  • [ASAP] Readily Reconfigurable Continuous-Stirred Tank Photochemical
           Reactor Platform

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      Authors: Daniel Francis; A. John Blacker, Nikil Kapur, Stephen P. Marsden
      Abstract: TOC GraphicOrganic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00428
      PubDate: Wed, 22 Dec 2021 05:00:00 GMT
       
  • [ASAP] Scale-Up and Development of Synthesis 2-Ethylhexyl Nitrate in
           Microreactor Using the Box–Behnken Design

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      Authors: Shuai Guo; Le-wu Zhan, Guang-kai Zhu, Xin-guang Wu, Bin-dong Li
      Abstract: TOC GraphicOrganic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00388
      PubDate: Wed, 22 Dec 2021 05:00:00 GMT
       
  • [ASAP] Employing Constant Rate Filtration To Assess Active Pharmaceutical
           Ingredient Washing Efficiency

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      Authors: Muhid Shahid; Chloé Faure, Sara Ottoboni, Leo Lue, Chris Price
      Abstract: TOC GraphicOrganic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00272
      PubDate: Tue, 21 Dec 2021 05:00:00 GMT
       
  • [ASAP] Breakage Study of the Urchinlike Crystal Clusters of Ibrutinib

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      Authors: Vít Zvoníček; Ondřej Stoklasa, Dan Trunov, Ivona Sedlářová, Tereza Boleslavská, Jiří Němeček, Miloslav Lhotka, Jiří Němeček, Pavel Žvátora, Miroslav Šoóš
      Abstract: TOC GraphicOrganic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00291
      PubDate: Mon, 20 Dec 2021 05:00:00 GMT
       
  • R)-α-Phenylethylamine&rft.title=Organic+Process+Research+&+Development&rft.issn=1083-6160&rft.date=2021&rft.volume=&rft.aulast=Cai&rft.aufirst=Baoqin&rft.au=Baoqin+Cai&rft.au=Jiyong+Wang,++Hu+Hu,++Sitong+Liu,++Chengxiao+Zhang,++Ying+Zhu,++Marco+Bocola,++Lei+Sun,++Yaoyao+Ji,++Ameng+Zhou,++Kuifang+He,++Qinli+Peng,++Xiao+Luo,++Ruimei+Hong,++Juanjuan+Wang,++Chuanyang+Shang,++Zikun+Wang,++Zhuhong+Yang,++Yong+Koy+Bong,++Thomas+Daussmann,++Haibin+Chen">[ASAP] Transaminase Engineering and Process Development for a Whole-Cell
           Neat Organic Process to Produce (R)-α-Phenylethylamine

    • Free pre-print version: Loading...

      Authors: Baoqin Cai; Jiyong Wang, Hu Hu, Sitong Liu, Chengxiao Zhang, Ying Zhu, Marco Bocola, Lei Sun, Yaoyao Ji, Ameng Zhou, Kuifang He, Qinli Peng, Xiao Luo, Ruimei Hong, Juanjuan Wang, Chuanyang Shang, Zikun Wang, Zhuhong Yang, Yong Koy Bong, Thomas Daussmann, Haibin Chen
      Abstract: TOC GraphicOrganic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00409
      PubDate: Fri, 17 Dec 2021 05:00:00 GMT
       
  • [ASAP] Development of a Commercial Process for Odalasvir

    • Free pre-print version: Loading...

      Authors: Duc N. Tran; Alexander Zhdanko, Santiago Barroso, Patrick Nieste, Ramdane Rahmani, Jan Holan, Roel Hoefnagels, Peter Reniers, Frederik Vermoortele, Stewart Duguid, Lionel Cazanave, Marek Figlus, Colin Muir, Alain Elliott, Peichao Zhao, Warren Paden, Cristina Hernandez Diaz, Stephen J. Bell, Akihiro Hashimoto, Avinash Phadke, Jason A. Wiles, Ilse Vogels, Vittorio Farina
      Abstract: TOC GraphicOrganic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00237
      PubDate: Wed, 15 Dec 2021 05:00:00 GMT
       
  • [ASAP] Synthesis of the C1–C13 Fragment of Eribulin on a Kilogram
           Scale

    • Free pre-print version: Loading...

      Authors: Seong Taek Kim; Yongseo Park, Namhyeon Kim, Jaeun Gu, Wongyoung Son, Jisu Hur, KangHee Lee, Areum Baek, Ju Young Song, U Bin Kim, Kee-Young Lee, Chang-Young Oh, Seokhwi Park, Hyunik Shin
      Abstract: TOC GraphicOrganic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00295
      PubDate: Tue, 14 Dec 2021 05:00:00 GMT
       
  • [ASAP] An Investigation into the Unexpected Corrosion of Nickel Alloy
           Vessels with Selectfluor

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      Authors: Tao Wang; Thomas P. Vickery, Donald Bachert, Rekha Gangam, Eric Margelefsky, Eric M. Phillips, Stephen M. Dalby, Wenjun Liu, Amanda Peterman, Kerstin Zawatzky, Ryan D. Cohen
      Abstract: TOC GraphicOrganic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00375
      PubDate: Mon, 13 Dec 2021 05:00:00 GMT
       
  • tert-butyl+Chloromethyl+Phosphate&rft.title=Organic+Process+Research+&+Development&rft.issn=1083-6160&rft.date=2021&rft.volume=&rft.aulast=Harper&rft.aufirst=Kaid&rft.au=Kaid+C.+Harper&rft.au=Russel+Klix,++Yu-Ming+Pu,++Jeremy+Henle,++Jianguo+Ji,++Yi-Yin+Ku">[ASAP] Mechanistic Evaluation and Solvent-Based Linear Free Energy
           Relationship in the Alkylation of ABT-199 Using Di-tert-butyl Chloromethyl
           Phosphate

    • Free pre-print version: Loading...

      Authors: Kaid C. Harper; Russel Klix, Yu-Ming Pu, Jeremy Henle, Jianguo Ji, Yi-Yin Ku
      Abstract: TOC GraphicOrganic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00363
      PubDate: Wed, 08 Dec 2021 05:00:00 GMT
       
  • [ASAP] Recommendations for Effective and Defendable Implementation of
           Quality by Design

    • Free pre-print version: Loading...

      Authors: Andrei A. Zlota
      Abstract: TOC GraphicOrganic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00265
      PubDate: Mon, 29 Nov 2021 05:00:00 GMT
       
  • [ASAP] Development of a High-Throughput Kinetics Protocol and Application
           to an Aza-Michael Reaction

    • Free pre-print version: Loading...

      Authors: Xiao Li; Anna L. Dunn
      Abstract: TOC GraphicOrganic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00213
      PubDate: Mon, 22 Nov 2021 05:00:00 GMT
       
  • [ASAP] Unconventional Synthetic Process of Fasudil Hydrochloride: Costly
           Homopiperazine Was Avoided

    • Free pre-print version: Loading...

      Authors: Jianhong Zhao; Dingding Wang, Wu-Lin Yang, Jinming Niu, Weiting Wu
      Abstract: TOC GraphicOrganic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00211
      PubDate: Mon, 22 Nov 2021 05:00:00 GMT
       
  • [ASAP] Removal of Alkyl Sulfonates Using DABCO

    • Free pre-print version: Loading...

      Authors: Kaitlyn Corazzata; Peter J. Rose, Shunyan Mo, Joseph Snodgrass, Alexander Langston, Elaine C. Lee
      Abstract: TOC GraphicOrganic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00335
      PubDate: Thu, 18 Nov 2021 05:00:00 GMT
       
  • [ASAP] Application of Machine Learning and Reaction Optimization for the
           Iterative Improvement of Enantioselectivity of Cinchona-Derived Phase
           Transfer Catalysts

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      Authors: Katrina W. Lexa; Kevin M. Belyk, Jeremy Henle, Bangping Xiang, Robert P. Sheridan, Scott E. Denmark, Rebecca T. Ruck, Edward C. Sherer
      Abstract: TOC GraphicOrganic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00155
      PubDate: Tue, 16 Nov 2021 05:00:00 GMT
       
  • [ASAP] Asymmetric Synthesis of the Cyclohexyl Fragment in RORγt Inhibitor
           

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      Authors: William P. Gallagher; John R. Coombs, Carlos A. Guerrero, Boguslaw M. Mudryk, Kishta Katipally, Candice L. Joe, Sanjeewa Rupasinghe, Jason Zhu, Francisco González-Bobes
      Abstract: TOC GraphicOrganic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00339
      PubDate: Tue, 16 Nov 2021 05:00:00 GMT
       
  • [ASAP] Manufacturing Process Development for Belzutifan, Part 5: A
           Streamlined Fluorination–Dynamic Kinetic Resolution Process

    • Free pre-print version: Loading...

      Authors: Tao Wang; Eric M. Phillips, Stephen M. Dalby, Eric Sirota, Stephanus Axnanda, C. Scott Shultz, Pratiq Patel, Jacob H. Waldman, Embarek Alwedi, Xiao Wang, Kerstin Zawatzky, Matthew Chow, Nilusha Padivitage, Mark Weisel, Michael Whittington, Jianjun Duan, Taotao Lu
      Abstract: TOC GraphicOrganic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00242
      PubDate: Mon, 15 Nov 2021 05:00:00 GMT
       
  • [ASAP] Manufacturing Process Development for Belzutifan, Part 6: Ensuring
           Scalability for a Deoxyfluorination Reaction

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      Authors: Michael Pirnot; Kevin Stone, Timothy J. Wright, David J. Lamberto, Jochen Schoell, Yu-hong Lam, Kerstin Zawatzky, Xiao Wang, Stephen M. Dalby, Adam J. Fine, Jonathan P. McMullen
      Abstract: TOC GraphicOrganic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00239
      PubDate: Fri, 12 Nov 2021 05:00:00 GMT
       
  • [ASAP] Manufacturing Process Development for Belzutifan, Part 2: A
           Continuous Flow Visible-Light-Induced Benzylic Bromination

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      Authors: Cecilia Bottecchia; François Lévesque, Jonathan P. McMullen, Yining Ji, Mikhail Reibarkh, Feng Peng, Lushi Tan, Glenn Spencer, Jarod Nappi, Dan Lehnherr, Karthik Narsimhan, Michael K. Wismer, Like Chen, Yipeng Lin, Stephen M. Dalby
      Abstract: TOC GraphicOrganic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00240
      PubDate: Thu, 11 Nov 2021 05:00:00 GMT
       
  • [ASAP] A Radical Addition Approach to a Heptafluoroisopropyl Substituted
           Arene, Combined with a Highly Diastereoselective Annulation Reaction To
           Synthesize the Tricyclic Core of BMS-986251

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      Authors: William P. Gallagher; John R. Coombs, Carlos A. Guerrero, Eric M. Simmons, Francisco González-Bobes
      Abstract: TOC GraphicOrganic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00338
      PubDate: Thu, 11 Nov 2021 05:00:00 GMT
       
  • [ASAP] Manufacturing Process Development for Belzutifan, Part 4: Nitrogen
           Flow Criticality for Transfer Hydrogenation Control

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      Authors: Nastaran Salehi Marzijarani; Adam J. Fine, Stephen M. Dalby, Rekha Gangam, Samiksha Poudyal, Taylor Behre, Anil R. Ekkati, Brittany M. Armstrong, C. Scott Shultz, Zachary E. X. Dance, Kevin Stone
      Abstract: TOC GraphicOrganic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00231
      PubDate: Wed, 10 Nov 2021 05:00:00 GMT
       
  • [ASAP] Manufacturing Process Development for Belzutifan, Part 3:
           Completing a Streamlined Through-Process with a Safe and Scalable
           Oxidation

    • Free pre-print version: Loading...

      Authors: Zhiwei Chen; Nastaran Salehi Marzijarani, Scott Quirie, Gregory F. Pirrone, Stephen M. Dalby, Tao Wang, Jungchul Kim, Feng Peng, Adam J. Fine
      Abstract: TOC GraphicOrganic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00232
      PubDate: Tue, 09 Nov 2021 05:00:00 GMT
       
  • [ASAP] Efficient Manufacturing Process for the Selective Estrogen Receptor
           Degrader GDC-9545 (Giredestrant) via a Crystallization-Driven
           Diastereoselective Pictet–Spengler Condensation

    • Free pre-print version: Loading...

      Authors: Jie Xu; Cheol K. Chung, Andrew McClory, Kyle A. Mack, Michael E. Dalziel, Alec Fettes, Kyle Clagg, Ngiap-Kie Lim, Georg Wuitschik, Christian Jenny, Laure Finet, Michael Kammerer, Haiming Zhang, Rémy Angelaud, Francis Gosselin
      Abstract: TOC GraphicOrganic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00263
      PubDate: Tue, 09 Nov 2021 05:00:00 GMT
       
  • [ASAP] Large-Scale Enantioselective Reduction of 2,3-Disubstituted
           Indenopyridine Enables a Practical Manufacturing Process for an 11β-HSD-1
           Inhibitor

    • Free pre-print version: Loading...

      Authors: Bo Qu; Xudong Wei, Xingzhong Zeng, Bing-Shiou Yang, Jean-Nicolas Desrosiers, Jolaine Savoie, Jun Wang, Maurice A. Marsini, Zhibin Li, Nizar Haddad, Jon C. Lorenz, Patrick Tielmann, Nora Maier, Jinhua J. Song, Chris H. Senanayake
      Abstract: TOC GraphicOrganic Process Research & Development
      DOI : 10.1021/acs.oprd.1c00290
      PubDate: Mon, 08 Nov 2021 05:00:00 GMT
       
  • [ASAP] Manufacturing Process Development for Belzutifan, Part 1: A Concise
           Synthesis of the Indanone Starting Material

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      Authors: Oliver T. Ring; Barry R. Hayter, Thomas O. Ronson, Lauren R. Agnew, Ian W. Ashworth, Janette Cherryman, Malcolm A. Y. Gall, Peter R. Hamilton, Phillip A. Inglesby, Martin F. Jones, Alex L. Lamacraft, Adam J. Leahy, David McKinney, Lucie Miller-Potucka, Lyn Powell, Okky D. Putra, Andrew J. Robbins, Simone Tomasi, Rosemary A. Wordsworth
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