Subjects -> CHEMISTRY (Total: 986 journals)
    - ANALYTICAL CHEMISTRY (59 journals)
    - CHEMISTRY (713 journals)
    - CRYSTALLOGRAPHY (23 journals)
    - ELECTROCHEMISTRY (28 journals)
    - INORGANIC CHEMISTRY (45 journals)
    - ORGANIC CHEMISTRY (47 journals)
    - PHYSICAL CHEMISTRY (71 journals)

ORGANIC CHEMISTRY (47 journals)

Showing 1 - 41 of 41 Journals sorted alphabetically
ACS Omega     Open Access   (Followers: 2)
Advances in Image and Video Processing     Open Access   (Followers: 18)
Advances in Physical Organic Chemistry     Full-text available via subscription   (Followers: 4)
Advances in Redox Research     Open Access   (Followers: 4)
American Journal of Organic Chemistry     Open Access   (Followers: 15)
Asian Journal of Organic Chemistry     Hybrid Journal   (Followers: 4)
Beilstein Journal of Organic Chemistry     Open Access   (Followers: 13)
Biochemia Medica     Open Access  
Current Organic Chemistry     Hybrid Journal   (Followers: 14)
Current Organic Synthesis     Hybrid Journal   (Followers: 12)
European Journal of Organic Chemistry     Hybrid Journal   (Followers: 59)
Herbal Medicine: Open Access     Open Access  
International Journal of Organic Chemistry     Open Access   (Followers: 9)
International Journal of Polymeric Materials     Hybrid Journal   (Followers: 6)
Journal of Bioactive and Compatible Polymers     Hybrid Journal   (Followers: 2)
Journal of Biomaterials Science, Polymer Edition     Hybrid Journal   (Followers: 9)
Journal of Organic Semiconductors     Open Access   (Followers: 6)
Journal of Peptide Science     Hybrid Journal   (Followers: 14)
Journal of Physical Organic Chemistry     Hybrid Journal   (Followers: 8)
Journal of Physiology and Biochemistry     Hybrid Journal   (Followers: 3)
Journal of Progressive Research in Chemistry     Open Access  
Journal of Proteins and Proteomics     Open Access   (Followers: 2)
Mini-Reviews in Organic Chemistry     Hybrid Journal   (Followers: 10)
Nigerian Journal of Chemical Research     Full-text available via subscription   (Followers: 1)
Open Journal of Organic Polymer Materials     Open Access   (Followers: 1)
Organic & Biomolecular Chemistry     Hybrid Journal   (Followers: 56)
Organic and Medicinal Chemistry Letters     Open Access   (Followers: 5)
Organic Chemistry : Current Research     Open Access   (Followers: 12)
Organic Chemistry Frontiers     Hybrid Journal   (Followers: 9)
Organic Chemistry International     Open Access   (Followers: 7)
Organic Geochemistry     Hybrid Journal   (Followers: 3)
Organic Letters     Hybrid Journal   (Followers: 92)
Organic Preparations and Procedures International: The New Journal for Organic Synthesis     Hybrid Journal   (Followers: 3)
Organic Process Research & Development     Hybrid Journal   (Followers: 32)
Progress in Organic Coatings     Hybrid Journal   (Followers: 7)
Reports in Organic Chemistry     Open Access   (Followers: 7)
Russian Journal of Organic Chemistry     Hybrid Journal   (Followers: 3)
Synthetic Communications: An International Journal for Rapid Communication of Synthetic Organic Chemistry     Hybrid Journal   (Followers: 31)
The Journal of Organic Chemistry     Hybrid Journal   (Followers: 135)
Vibrational Spectroscopy     Hybrid Journal   (Followers: 11)
World Journal of Organic Chemistry     Open Access   (Followers: 5)
Similar Journals
Journal Cover
Organic & Biomolecular Chemistry
Journal Prestige (SJR): 1.281
Citation Impact (citeScore): 3
Number of Followers: 56  
 
  Hybrid Journal Hybrid journal (It can contain Open Access articles)
ISSN (Print) 1477-0520 - ISSN (Online) 1477-0539
Published by RSC Homepage  [49 journals]
  • Pd and photoredox dual catalysis assisted decarboxylative
           ortho-benzoylation of N-phenyl-7-azaindoles

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02338A, PaperShruti Rajput, Ramandeep Kaur, Nidhi Jain
      Directing group assisted decarboxylative ortho-benzoylation of N-aryl-7-azaindoles with α-keto acids has been achieved by synergistic visible light promoted photoredox and palladium catalysis. The approach tenders rapid entry to aryl ketone...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Ligand Centered Redox Enabled Sustainable Synthesis of Triazines and
           Pyrimidines Using A Zinc-Stabilized Azo-Anion Radical Catalyst

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02428K, PaperSiuli Das, Rakesh Mondal, Amit Kumar Guin, Nanda D Paul
      Herein, we report ligand-centered redox controlled Zn(II)-catalyzed multicomponent approaches for synthesizing pyrimidines and triazines. Taking advantage of the ligand-centered redox events, using a well-defined Zn(II)-catalyst (1a) bearing (E)-2-((4-chlorophenyl)diazenyl)-1,10-phenanthroline (L1a) as...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Hydrogenation of cage-opened C60 derivatives mediated by frustrated Lewis
           pairs

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Advance Article

      DOI : 10.1039/D1OB02316K, CommunicationYoshifumi Hashikawa, Yasujiro Murata
      Multiply-carbonylated fullerene derivatives were found to work as one component in frustrated Lewis pairs which caused an Si–H bond activation in the presence of B(C6F5)3, leading to the carbonyl hydrogenation in up to 99% yield.
      To cite this article before page numbers are assigned, use the
      DOI form of citation above.
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Dienylation of N-benzoylhydrazones with CF3-substituted
           Homoallenylboronates in Water

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02335G, CommunicationWei-Wei Ma, Chao Yang, Qiang Xie, Yun-He Xu
      A convenient method for the dienylation of N-benzoylhydrazones was developed in water without any inert gas protection. The 2-methylamino-1,3-diene derivatives could be produced in water without additional catalyst and additive....
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Synthetic and biosynthetic methods for selective cyclisations of 4,5-epoxy
           alcohols to tetrahydropyrans

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Advance Article

      DOI : 10.1039/D1OB01905H, Review ArticleOpen Access Open Access Creative Commons Licence  This article is licensed under a Creative Commons Attribution 3.0 Unported Licence.James I. Bowen, Luoyi Wang, Matthew P. Crump, Christine L. Willis
      In this review, methods for the selective intramolecular epoxide ring opening (IERO) of 4,5-epoxy-alcohols are discussed as well as biosynthetic pathways to tetrahydropyran-containing natural products which utilise IERO reactions.
      To cite this article before page numbers are assigned, use the
      DOI form of citation above.
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Visible-light-mediated tandem phosphorylation/cyclization for the
           synthesis of phosphorylated oxindoles

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02486H, CommunicationLiu-Liang Mao, An-Xi Zhou, Xian-Hong Zhu, Li-Xia Quan, Fayun Chen, Jie-Ping Wan, Yinlong Lai
      The visible-light-mediated tandem phosphorylation/cyclization of Narylacrylamides with H-phosphine oxides has been developed for the synthesis of phosphorylated oxindoles. This efficient and facile process was useful for the construction of C−P...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Development of a single-step fluorogenic sirtuin assay and its
           applications for high-throughput screening

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02347K, PaperPan Wang, Di Chen, Jianxiong An, Shu-xian Lin, Ting Liu, Yan Li, Lei Chen, Bin He
      Sirtuins (SIRTs) are a class of nicotinamide adenine dinucleotide (NAD+)-dependent histone deacetylases. Since SIRTs have different subcellular locations and different preferences for deacylation activity, SIRTs are not only highly gaining...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • The supramolecular chemistry of anions

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Advance Article

      DOI : 10.1039/D1OB90183D, EditorialKatrina (Kate) A. Jolliffe, Philip A. Gale
      Guest editors Katrina Jolliffe and Philip Gale introduce the Organic & Biomolecular Chemistry themed collection on the supramolecular chemistry of anions.
      To cite this article before page numbers are assigned, use the
      DOI form of citation above.
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Tetradentate halogen bonding macrocyclic anion receptor inspired by the
           “Texas-sized” molecular box

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02381K, CommunicationTian Zhao, Vincent Lynch, Jonathan L. Sessler
      Inspired by the tetracationic “Texas-sized” molecular box, a neutral analogue containing four iodotriazole halogen bond-promoting subunits (“Ibox”) was synthesized. This new macrocycle was prepared by means of azide-alkyne click chemistry....
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Correction: The kinetic resolution of oxazinones by alcoholysis: access to
           orthogonally protected β-amino acids

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Advance Article

      DOI : 10.1039/D1OB90184B, CorrectionOpen Access Open Access Creative Commons Licence  This article is licensed under a Creative Commons Attribution 3.0 Unported Licence.Sarah A. Cronin, Stephen J. Connon
      To cite this article before page numbers are assigned, use the
      DOI form of citation above.
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Enantioselective “Clip-Cycle” Synthesis of Di-, Tri- and Spiro-
           Substituted Tetrahydropyrans

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D2OB00023G, Communication Khadra Alomari, N. Sai Pavan Chakravarthy, Bastien Duchadeaau, Kristaps Ermanis, Paul Clarke
      ω-Unsaturated alcohols were “clipped” via alkene metathesis to a thioester activating group, which was followed by a chiral phosphoric acid catalyzed intramolecular oxa-Michael cyclization to yield tetrahydropyrans and spiro-tetrahydropyrans with...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Discovery of 13,15-nor-Polycyclic Polyprenylated Acylphloroglucinols from
           Hypericum longistylum with Anti-Inflammatory Activity

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02107A, PaperZhengyi Shi, Hong Hu, Yi Guo, Yulin Duan, Yeting Zhang, Bo Tao, Pengfei Bu, Weiguang Sun, Changxing Qi, Yonghui Zhang
      Spihyperglucinols A (1) and B (2), the first 13,15-nor-polycyclic polyprenylated acylphloroglucinols (PPAPs) featuring a 7/6/5 tricyclic ring system based on an unexpected bicyclo[3.2.2]nonane core, along with three new congeners, spihyperglucinols...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Metal-Free Alkylation of Quinoxalinones with Aryl Alkyl ketones

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02260A, CommunicationXinya Liu, Zhuangzhuang Guo, Yanpeng Liu, Xiaoyu Chen, Jingya Li, Dapeng Zou, Yangjie Wu, Yusheng Wu
      The first metal-free method for alkylation of quinoxalinones using cheap and stable aryl alkyl ketones as nucleophilic alkylation reagents is reported. This strategy greatly broadens the application channels of aryl...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Azomethine ylide cycloaddition of 1,3-dienyl esters: highly regio- and
           diastereoselective synthesis of functionalized pyrrolidinochromenes

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Advance Article

      DOI : 10.1039/D1OB02042K, CommunicationManickam Bakthadoss, Mohammad Mushaf, Vishal Agarwal, Tadiparthi Thirupathi Reddy, Duddu S. Sharada
      Highly regio- and diastereoselective synthesis of functionalized pyrrolidinochromenes via azomethine ylide cycloaddition reaction has been developed with excellent yields and wide substrate scope.
      To cite this article before page numbers are assigned, use the
      DOI form of citation above.
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Light-responsive molecular switch based on cucurbit[7]uril and
           1,1'-bis(benzyl)-4-[2-(4-pyridyl)-vinyl]-pyridinium dibromide displaying
           white light emission

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02420E, Paperqin wang, Kun Zhang, Rui-Lian Lin, Wenqi Sun, Mingfu Ye, Xin Xiao, Jingxin Liu
      By using 1H NMR, ESI-MS and UV spectra, novel light-responsive molecular switch constructed by 1,1’-bis(benzyl)-4-[2-(4-pyridyl)-vinyl]-pyridinium (12+) and cucurbit[7]uril (Q[7]) is demonstrated. The E- to Z-isomerization of double bond in 12+...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Reaction-based fluorescence probes for “turn on” sensing
           fluoride ions

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02324A, CommunicationWen-Ying He, Ning Liu, Xu Jiang, Yan-Zhen Zheng, Zhi-Wei Lin, Jiang-Shan Shen
      Introducing a weak covalent bond into an originally highly fluorescent molecule to create a non-fluorescent probe is able to afford a new way to detect some neucleophilic targets with enhanced...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Magnesium dicarboxylates promoted prenylation of phenolics that was
           elaborated for the total synthesis of icaritin

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02228H, PaperJichao Zhang, Wei Xiong, Yongju Wen, Xuewen Fu, Xiaoxia Lu, Guo-Lin Zhang, Chun Wang
      The prenylation of phenolic substrates promoted by Magnesium dicarboxylates was developed. Investigation of the scope demonstrated that substrats with electron-donating group(s) gave better yield than those of electron-withdrawing group(s). Although...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Pd-catalyzed desulfitative arylation of olefins by N-methoxysulfonamide

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02360H, PaperSubhadra Ojha, Niranjan Panda
      A novel Pd-catalyzed protocol desulfitative Heck type reaction of N-methoxy aryl sulfonamides with alkenes was reported. The cross-coupling reaction was performed successfully with a variety of olefins to obtainaryl alkenes....
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Rh(III)-catalyzed annulated coupling of sulfoxonium ylides and iodonium
           ylides: a rapid access to isocoumarins

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02273C, PaperChuanliu Yin, Lianghao Li, Chuanming Yu
      Direct synthesis of isocoumarin skeletons has been realized through Rh(III)-Catalyzed [3 + 3] annulation of sulfoxonium ylides and iodonium carbenes. The synthetic protocol constructed efficiently with the broad functional group...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • An iron-catalyzed domino reaction of donor–acceptor cyclopropanes: a
           diastereoselective approach towards diversely functionalized
           pyrrolo-quinazolines

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Advance Article

      DOI : 10.1039/D1OB02215F, PaperSamiran Dhara, Subhadeep Ghosh, Asish R. Das
      An expeditious synthetic route to access functionalized pyrrolo[2,1-b]quinazoline scaffolds has been achieved via domino ring opening cyclization (DROC) reactions of donor–acceptor (D–A) cyclopropanes and 2-amino(methyl)aniline derivatives.
      To cite this article before page numbers are assigned, use the
      DOI form of citation above.
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Copper–Catalyzed Thiocarbonylation and Thiolation of Alkyl Iodides

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D2OB00008C, CommunicationYahui Li, Qingqiang Tian, Rongjing Sun
      In the present study, an efficient Cu-catalyzed transthiolation of alkyl iodides has been developed. Notably, in the presence of CO, thioesters could also be obtained with copper and cobalt as...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Cu-Catalyzed alkylation–cyanation type difunctionalization of styrenes
           with aliphatic aldehydes and TMSCN via decarbonylation

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02376D, PaperYu-Ling Zhou, Jun-Jia Chen, Jing Cheng, Luo Yang
      A copper-catalyzed decarbonylative alkylation–cyanation of styrene derivatives with aliphatic aldehydes and trimethylsilyl cyanide to provide chain elongated nitriles is reported. Using TBHP as oxidant and free radical initiator, the reaction...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Deoxy sugars. General methods for carbohydrate deoxygenation and
           glycosidation

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Advance Article

      DOI : 10.1039/D1OB02001C, Review ArticleCarla Marino, Andrea V. Bordoni
      The methods for the synthesis of deoxy sugars, involving deoxygenation and glycosidation, give access to useful molecules for multiple purposes.
      To cite this article before page numbers are assigned, use the
      DOI form of citation above.
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Iodine-Catalyzed Oxidative Annulation: Facile Synthesis of
           

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02436A, PaperXin-Ke Zhang, Xiao-Yu Miao, Yu Zhou, Yu-Mei Wang, Ying-Chun Song, Hang Liu, Yi-Lu Xiong, Ling-Yu Li, An-Xin Wu, Yan-Ping Zhu
      An iodine-catalytic methyl azaarenes sp3 C-H functionalization has been developed for synthesis of a seven-membered O-heterocyclic architecture containing three different heterocyclic aromatic hydrocarbons. This method can be applied to a...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Transaminases as suitable catalysts for the synthesis of enantiopure
           β,β-difluoroamines

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02346B, CommunicationMarina García-Ramos, Iván Lavandera
      Transaminases have demonstrated the ability to catalyze the amination of a series of aliphatic and (hetero)aromatic α,α-difluorinated ketones with high stereoselectivity, thus providing the corresponding β,β-difluoroamines in high isolated yields...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • The Role of Acetylated Cyclooxygenase-2 in the Biosynthesis of Resolvin
           Precursors Derived from Eicosapentaenoic Acid

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB01932E, PaperAnna Cebrián-Prats, Alexandre Pinto, Àngels González-Lafont, Pedro Alexandrino Fernandes, José M Lluch
      Specialized pro-resolving lipid mediators (SPMs) are natural bioactive agents actively involved in inflammation resolution. SPMs act when uncontrolled inflammatory processes are developed, for instance, in patients of COVID-19 or other...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • NHC-Catalyzed [4+2] Annulations of Allenoates and 2,3-Dioxopyrrolidine
           Derivatives

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02180J, PaperXue Song, Yangxu Chen, Fangfang Lu, Kai Zhang, Chenxia Yu, Tuanjie Li, Changsheng Yao
      A facile NHC-catalyzed [2+4] annulation of allenoates with 2,3-dioxypyrrolidine derivatives was discovered, which paved a new avenue to the construction of highly substituted pyranopyrrole with moderate to good yields, high...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Constructing Firefly Luciferin Bioluminescence Probes for in Vivo Imaging

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB01940F, Review ArticleXingye Yang, Xiaojun Qin, Huimin Ji, Lupei Du, Minyong Li
      Bioluminescence imaging (BLI) is a widely applied visual approach for real-time detecting many physiological and pathological processes in a variety of biological systems. Based on the caged strategy, lots of...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Diazaborines Oxidize Slowly with H2O2 but Rapidly with Peroxynitrite in
           Aqueous Buffer

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB01668G, CommunicationJack G. Haggett, Gun Su Han, Angela R. Moser, Julian V.A. Golzwarden, Shubham Vyas, Dylan W Domaille
      Reactive oxygen species (ROS) such as H2O2 and peroxynitrite (ONOO-) oxidize arylboronic acids to their corresponding phenols. When used in molecular imaging probes and in ROS-responsive molecules, however, simple arylboronic...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Cyclobutane Based “Overbred Intermediates” and it’s Exploration in
           Organic Synthesis

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02361F, Review ArticleSamik Nanda, Monosij Nandy, Swagata Das
      “Overbred intermediates” are being used in organic synthesis for a long time, but these intermediates are not categorized as overbred intermediate, this name was given recently in Hoffman's book “Elements...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Electroreductive synthesis of polyfunctionalized pyridin-2-ones from
           acetoacetanilides and carbon disulfide with oxygen evolution

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02379A, CommunicationLichun Xu, Zhongxiao Ma, Xi Hu, Xin Zhang, Shulin Gao, Deqiang Liang, Baoling Wang, Weili Li, Yanni Li
      A chemical reductant or a sacrificial electron donor is required in any reduction reaction, generally resulting in undesired chemical wastes. Herein, we report a reductant-free reductive [3+2+1] annulation of β-keto...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • An experimental and computational study for a Pd(II) catalysed
           hydroboration and reductive amination reaction of carbonyl compounds

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02339J, PaperTarun Kanti Panda, Shreya Mahato, Parveen Rawal, Ajitaro Devadkar , Mayank Joshi, Angshuman Roychoudhury, Bhaskar Biswas, Puneet Gupta
      We report the synthesis, characterisation, and catalytic application of a palladium (II) complex [(4-{1,2-C6H4(N=CH-C6H4O)2}Pd] (1) supported by a dianionic salen ligand [1,2-C6H4(N=CH-C6H4O)2]2- (L) as a molecular pre-catalyst for the hydroboration...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • On the Mechanism of the Dyotropic Expansion of Hydrindanes into Decalins

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02150H, PaperCarlos Silva Lopez, Yagamare Fall, Generosa Gómez, Olalla Nieto Faza, Hugo Santalla
      A combined computational/experimental approach has revealed key mechanistic aspects in a recently reported dyotropic expansion of hydrindanes into decalins. While computer simulations had already anticipated the need for acid catalysis...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Structure-Affinity Relationships of Reversible Proline Analog Inhibitors
           Targeting Proline Dehydrogenase

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02328D, PaperAlexandra Bogner, John Tanner
      Proline dehydrogenase (PRODH) catalyzes the first step of proline catabolism, the FAD-dependent oxidation of L-proline to Δ1-pyrroline-5-carboxylate. PRODH plays a central role in the metabolic rewiring of cancer cells, which...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • A Metal-Free Strategy for the Cross-Dehydrogenative Coupling of the 1,
           3-Dicarbonyl Compounds with 2-Methoxyethanol

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02290C, PaperVishal Suresh Kudale, Zheng Sheng, Sheng-Hua Huang, Yu-Lun Chang, Jeh-Jeng Wang
      Here, we report a metal-free approach for the construction of methylene-bridged bis-1,3-dicarbonyl compounds via cross-dehydrogenative coupling of 1,3-dicarbonyl compounds with 2-methoxyethanol. In addition, we have extended this methodology to synthesize...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Visible-light-mediated regioselective synthesis of novel
           thiazolo[3,2-b][1,2,4]triazoles: advantageous synthetic application of
           aqueous conditions

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Advance Article

      DOI : 10.1039/D1OB02194J, PaperRanjana Aggarwal, Mona Hooda, Prince Kumar, Mari Carmen Torralba
      A regioselective synthesis of novel thiazolo[3,2-b][1,2,4]triazoles has been established via a visible-light-facilitated reaction of unsymmetrical α-bromodiketones with 3-mercapto[1,2,4]triazoles under aqueous conditions.
      To cite this article before page numbers are assigned, use the
      DOI form of citation above.
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Electrocatalysis as a key strategy for the total synthesis of natural
           products

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Advance Article

      DOI : 10.1039/D1OB02115J, Review ArticleMintu Munda, Sovan Niyogi, Kundan Shaw, Sourav Kundu, Rhituparna Nandi, Alakesh Bisai
      This review provides an overview of the total syntheses of structurally intriguing natural products in which electrochemical processes play an important role as a key methodology.
      To cite this article before page numbers are assigned, use the
      DOI form of citation above.
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Unexpected ring opening of pyrazolines with activated alkynes: synthesis
           of 1H-pyrazole-4,5-dicarboxylates and chromenopyrazolecarboxylates

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, 20,334-338

      DOI : 10.1039/D1OB01727F, CommunicationSai Teja Kolla, Nageswara Rao Rayala, Balasubramanian Sridhar, China Raju Bhimapaka
      1H-Pyrazole-4,5-dicarboxylates and chromenopyrazolecarboxylates were prepared by the reaction of pyrazolines with activated alkynes under neat conditions without a catalyst for the first time.
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Metal–ligand cooperative approaches in homogeneous catalysis using
           transition metal complex catalysts of redox noninnocent ligands

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, 20,296-328

      DOI : 10.1039/D1OB01153G, Review ArticleRakesh Mondal, Amit Kumar Guin, Gargi Chakraborty, Nanda D. Paul
      Catalysis offers a straightforward route to prepare various value-added molecules starting from readily available raw materials.
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Brønsted acid-catalyzed enantioselective addition of 1,3-diones to in
           situ generated N-acyl ketimines

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, 20,410-414

      DOI : 10.1039/D1OB02162A, PaperMilon M. Sadhu, Sumit K. Ray, Rajshekhar A. Unhale, Vinod K. Singh
      A Brønsted acid-catalyzed enantioselective addition of 1,3-diones to in situ generated N-acyl ketimines has been developed. Various dicarbonyl-substituted chiral isoindolinones were achieved with up to 98% yields and up to 95% enantioselectivities.
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Molecular tetrominoes: selective masking of the donor π-face to control
           the configuration of donor–acceptor complexes

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, 20,375-386

      DOI : 10.1039/D1OB02293H, PaperJenna L. Sartucci, Arindam Maity, Manikandan Mohanan, Jeffery Bertke, Miklos Kertesz, Nagarjuna Gavvalapalli
      π-face masking opens up a new pathway to control the location of acceptor along the donor backbone and consequently donor–acceptor binding interaction strength and percentage of acceptor ionization.
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • The influence of α-coordinating groups of aldehydes on E/Z-selectivity
           and the use of quaternary ammonium counter ions for enhanced E-selectivity
           in the Julia–Kocienski reaction

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, 20,329-333

      DOI : 10.1039/D1OB02126E, CommunicationMintu Rehman, Sravya Surendran, Nagendra Siddavatam, Goreti Rajendar
      Enhanced E-selectivity of olefins in Julia-Kocienski reaction of aldehydes with α-coordinating groups is demonstrated using TBAB. A systematic study is presented to show the chelation effect and size of the protecting group on E/Z-selectivity.
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Studies directed toward the synthesis of hedycoropyrans: total synthesis
           of des-hydroxy (−)-hedycoropyran B (ent-rhoiptelol B)

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, 20,444-463

      DOI : 10.1039/D1OB01972D, PaperPriyanka Kataria, Rajesh Nomula, Ravindar Kontham
      Studies directed towards the stereoselective synthesis of the diarylheptanoid-derived natural products hedycoropyrans leading to the total synthesis of (−)-hedycoropyran B (ent-rhoiptelol B) are presented.
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Cascade synthesis of indolizines and pyrrolo[1,2-a]pyrazines from
           2-formyl-1-propargylpyrroles

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, 20,396-409

      DOI : 10.1039/D1OB01839F, PaperCarlos H. Escalante, Fernando A. Carmona-Hernández, Alberto Hernández-López, Eder I. Martínez-Mora, Francisco Delgado, Joaquín Tamariz
      A cascade reaction of 2-formyl-N-propargylpyrroles or N-allenyl-2-formylpyrroles with active methylene compounds and ammonium acetate provides indolizines and pyrrolo[1,2-a]pyrazines, respectively.
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Recent advances in palladium-catalyzed C(sp3)/C(sp2)–H bond
           functionalizations: access to C-branched glycosides

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, 20,264-281

      DOI : 10.1039/D1OB02142G, Review ArticleZanjila Azeem, Pintu Kumar Mandal
      This review summarises recent developments in palladium-catalyzed directed and nondirected C–H functionalization approaches to access C-branched aryl/alkenyl/alkyl glycosides with reaction characteristics and proposed mechanisms.
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Recent developments in the synthesis of nitrogen-containing heterocycles
           from β-aminovinyl esters/ketones as CC–N donors

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, 20,282-295

      DOI : 10.1039/D1OB01998H, Review ArticleXiao-Feng Xia, Yan-Ning Niu
      The synthesis of nitrogen-containing heterocycles from β-aminovinyl esters(ketones) was reviewed according to the classification of the final heterocycle synthesis.
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Ligand-free copper-catalyzed borylative defluorination: access to
           gem-difluoroallyl boronic acid derivatives

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, 20,366-374

      DOI : 10.1039/D1OB01533H, PaperAshley M. Gates, Swetha Jos, Webster L. Santos
      We report a ligand-free copper-catalyzed β-borylation, defluorination of β-substituted, α-trifluoromethyl-α,β-unsaturated esters.
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Cross Dehydrogenation Coupling Reaction of Purine Derivatives with
           Thioethers

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02353E, PaperXinjie Li, Peng Qi, Hongguang Du
      A metal-free cross-dehydrogenation coupling method was established to synthesize N9 alkylated purine derivatives. Using PhI(OAc)2 as oxidants, versatile thioethers were successfully employed as alkylation reagents, Under optimized conditions, a variety...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Antifungal mono- and dimeric nitrogenous bisabolene derivatives from a
           sponge in the order Bubarida from Futuna Islands

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02297K, PaperMaría Miguel-Gordo, Maggie Reddy, Pilar Sanchez, Jordan Buckley, Thomas Mackenzie, Laurence Jennings, Fernando Reyes, Kevin Calabro, Olivier P Thomas
      An abundant sponge of the order Bubarida was selected for further chemical investigation following biological and chemical screening of sponges collected from Futuna Islands in the Indo-Pacific. Ten new nitrogenous...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • A base-mediated aerobic oxidative synthesis of cyclopent-2-enols
           derivatives from doubly activated cyclopropanes and substituted
           acetonitriles

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02155A, PaperXiao Dan Han, Gao Liang Peng, Wei Xiong, Ran Gan, Jian Ping Fu, lei wu, Zhong Sheng Tang, ju wu hu, hui bin wang
      We report here that polysubstituted cyclopent-2-enols can be constructed by the one-pot reaction of doubly activated cyclopropanes and ɑ-EWG substituted acetonitriles under mild basic conditions via a domino-ring-opening-cyclization /deacylation/oxidation sequence....
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Copper-Promoted Difunctionalization of Unactivated Alkenes with Silanes

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02318G, CommunicationYingying Xue, Zhuangzhuang Guo, Xiaoyu Chen, Jingya Li, Dapeng Zou, Yangjie Wu, Yusheng Wu
      An efficient copper-catalyzed cascade difunctionalization of N-allyl anilines toward the synthesis of silylated indolines using commercially available silanes has been reported. This strategy provides a new avenue for the synthesis...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Construction of azaspirocyclic skeletons mediated by the carbonyl of
           Weinreb amide: formal total synthesis of (±)-cephalotaxine

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02304G, CommunicationJian Zhang, Jianyin Liu, Yuxue Fan, Huili Ding, Tianfu Liu, Shanshan Li, Minghua Jiang, Lu Liu
      Facile stevens rearrangement of the Weinreb amide and the subsequent key steps mediated by the carbonyl of Weinreb amide led to the construction of azaspirocyclic skeletons of some typical alkaloids....
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Enantioselective organocatalytic syntheses of α-selenated α- and
           β-amino acid derivatives

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02235K, PaperOpen Access Open Access Creative Commons Licence  This article is licensed under a Creative Commons Attribution 3.0 Unported Licence.Victoria Haider, Paul Zebrowski, Jessica Michalke, Uwe Monkowius, Mario Waser
      Selenium-containing amino acids are valuable targets but methods for the stereoselective α-selenation of simple amino acid precursors are rare. We herein report the enantioselective electrophilic α-selenation of azlactones (masked α-amino...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Radiosynthesis and Evaluation of A Fluorine-18 Radiotracer [18F]FS1P1 for
           Imaging Sphingosine-1-Phosphate Receptor 1

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02225C, PaperLin Qiu, Hao Jiang, Yanbo Yu, Jiwei Gu, Jinzhi Wang, Haiyang Zhao, Tianyu Huang, Robert J Gropler, Robyn Klein, Joel S Perlmutter, Zhude Tu
      Assessment of Sphingosine-1-phosphate receptor 1 (S1PR1) expression could be a unique tool to determine the neuroinflammatory status for central nervous system (CNS) disorders. Our preclinical results indicate that PET imaging...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Synthesis and anti-tumor activity evaluation of salinomycin
           C20-O-alkyl/benzyl oximes derivatives

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02292J, PaperBO LI, Jun Wu, Lei Tang, Xu Lian, Zhongwen Li, Wenfang Duan, Tong Qing, Xintong Zhao, Yuhua Hu, Chi Zhang, Tianlei Li, Jie Hao, Wenxuan Zhang, Jihong Zhang, Song Wu
      Seventeen C20-O-alkyl/benzyl oximes derivatives were synthesized in concise and effective method. Most of these derivatives showed tens to several hundreds nanomolar IC50 values against HT-29 colorectal, HGC-27 gastric and MDA-MB-231...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Deuterium Labelling to Extract Local Stereochemical Information by VCD
           Spectroscopy in C-D Stretching Region: A Case Study of Sugars

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02317A, PaperMohamad Zarif Mohd Zubir, Nurul Fajry Maulida, Yoshihiro Abe, Yuta Nakamura, Mariam Abdelrasoul, Tohru Taniguchi, Kenji Monde
      Stereochemical elucidation of molecules with multiple chiral centers is difficult. Even with VCD spectroscopy, excluding all but one diastereomeric structural candidates is challenging because stereochemical inversion of one chiral center...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Squaramide‐catalysed asymmetric cascade Michael addition/acyl transfer
           reaction between unsaturated benzothiophenones and α-nitroketones

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02217B, PaperCheng Niu, Da-Ming Du
      An efficient and practical organocatalytic asymmetric strategy was developed using unsaturated benzothiophenones and α‐nitroketones catalysed by bifunctional squaramide via Michael addition and acyl transfer steps. A broad range of chiral...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Cross-conjugation controls the stabilities and photophysical properties of
           heteroazoarene photoswitches

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02026A, PaperDaniel Adrion, Steven A. Lopez
      Azoarene photoswitches are versatile molecules that interconvert from their E-isomer to their Z-isomer with light. Azobenzene is a prototypical photoswitch but its derivatives can be poorly suited for in vivo...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • N-alkylation of organonitrogen compounds catalyzed by methylene-linked
           bis-NHC half-sandwich ruthenium complexes

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02214H, PaperZakaria Moutaoukil, Emmanuel Serrano-Diez, I. Gonzalez Collado, Manuel Jimenez-Tenorio, José Manuel Botubol-Ares
      An efficient ruthenium-catalyzed N-alkylation of amines, amides and sulfonamides has been developed employing novel pentamethylcyclopentadienylruthenium (II) complexes bearing the methylene linked bis(NHC) ligand bis(3-methylimidazol-2-ylidene)methane. The acetonitrile complex 2 has proven...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Preparation of Nitriles from Aldehydes using Ammonium Persulfate by means
           of a Nitroxide-Catalysed Oxidative Functionalisation Reaction

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02187G, PaperArturo Leon Sandoval, Fabrizio Politano, Mason Witko, Nicholas E. Leadbeater
      A methodology for the preparation of nitriles from aldehydes by means of an oxidative functionalisation reaction is reported. It employs employs ammonium persulfate as the primary oxidant and the nitrogen...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Silver Salt Enabled H/D Exchange at β Position of Thiophene Rings:
           Synthesis of Fully Deuterated Thiophene derivatives

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02285G, CommunicationFei-fei Sheng, En-Ci Li, Jing-Wen Bai, Cai-Xia Wang, Guang-Qi Hu, Kai-Hui Liu, Zhengyi Sun, Kang Shen, Honghai Zhang
      We disclose a silver catalyzed H/D exchange reaction, which can introduce deuterium atom at β position of thiophene rings without the assisstance of any coordinating groups. The advantages of this...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Evaluation of DNA-mediated electron transfer using a hole-trapping
           nucleobase under crowded conditions

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB01669E, CommunicationYuuki Taketomi, Yuuki Yamaguchi, Shunsuke Sakurai, Makiko Tanaka
      The effects of a crowded environment on DNA-mediated electron transfer were evaluated using a pyrene-modified oligonucleotide containing a hole-trapping nucleobase in poly(ethylene glycol) mixed solutions. Rapid decompositions of hole-trapping bases...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Rhodium(III)-Catalyzed Cascade C−H Functionalization/Annulation of
           Sulfoximines with Iodonium Ylides for the Synthesis of
           Cyclohexanone-1,2-benzothiazines

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02110A, PaperLu Chen, Zhichao Wang, Yangyang Wang, Liqiang Hao, Xiaobo Xu, Gao-Rong Wu, Yafei Ji
      A highly efficient Rh(III)-catalyzed cascade C−H activation/annulation of sulfoximines with iodonium ylides under metal-oxidant-free conditions has been reported. The fused cyclohexanone-1,2-benzothiazine scaffold is readily achieved with a one-pot process in...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Recent developments in the utility of saturated azaheterocycles in
           peptidomimetics

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB01329G, Review ArticleManish Kumar Singh, Mahesh K Lakshman
      To large extent, the physical and chemical properties of peptidomimetic molecules are dictated by the integrated heterocyclic scaffolds they contain. Heterocyclic moieties are introduced into a majority of peptide-mimicking molecules...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Anion binding to a cationic europium(III) probe enables the first
           real-time assay of heparan sulfotransferase activity

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Advance Article

      DOI : 10.1039/D1OB02071D, PaperOpen Access Open Access Creative Commons Licence  This article is licensed under a Creative Commons Attribution 3.0 Unported Licence.Simon Wheeler, Colum Breen, Yong Li, Sarah H. Hewitt, Erin Robertson, Edwin A. Yates, Igor L. Barsukov, David G. Fernig, Stephen J. Butler
      We present a new luminescent europium(III)-based anion receptor that binds to PAP (adenosine-3′,5′-diphosphate). The increased emission intensity and lifetime of the receptor-PAP complex was used to develop the first real-time assay of heparan sulfotransferase activity.
      To cite this article before page numbers are assigned, use the
      DOI form of citation above.
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • A DFT examination of the role of proximal boron functionalities in the
           S-alkylation of sulfenic acid anions

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Advance Article

      DOI : 10.1039/D1OB02083H, PaperAndrew G. Durant, Eric A. Nicol, Brandon M. McInnes, Adrian L. Schwan
      DFT modelling predicts proximal boron groups can accelerate sulfenate alkylation reactions, depending on boron substituents and boron distance from the reaction site.
      To cite this article before page numbers are assigned, use the
      DOI form of citation above.
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • (±)-Usphenethylones A−C, three pairs of heterodimeric polyketide
           enantiomers from Aspergillus ustus 3.3904

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02006D, PaperHanli Ruan, Xiaogang Peng, Shuang Zhou, Junjun Liu, Ying Gao, Jinling Chang
      Three pairs of novel heterodimeric polyketide enantiomers, (±)-usphenethylones A−C (1−3), were isolated from the culture extract of Aspergillus ustus 3.3904. Compounds 1−3 represent two unique heterodimerization patterns of a phenethyl...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Controlling chirality in the synthesis of 4 + 4 diastereomeric amine
           macrocycles derived from trans-1,2-diaminocyclopentane and
           2,6-diformylpyridine.

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02410H, PaperDominka Fedorowicz, Sylwia Banach, Patrycja Koza, Rafał Frydrych, Katarzyna Ślepokura, Janusz Gregoliński
      A few suitably long dialdehyde and primary diamine building blocks of a predetermined chirality have been designed and synthesized to enable controlled and efficient synthesis of all 6 possible diastereomers...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • α-Functionalization of ketones promoted by sunlight and heterogeneous
           catalysis in the aqueous phase

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02249K, CommunicationLei He, Chenfeng Liang, Ya-Ni Ouyang, Lin Li, Yirui Guo, Peng-Fei Zhang, Wanmei Li
      Herein, a protocol that combined the heterogeneous catalysis and solar photocatalysis for the regioselective α-substitution of asymmetric ketones with quinoxalinones has been reported. The result indicates that the reaction is...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Synthesis of Broad-Specificity Activity-Based Probes for
           Exo-β-Mannosidases

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02287C, PaperOpen Access Open Access Creative Commons Licence  This article is licensed under a Creative Commons Attribution 3.0 Unported Licence.Nicholas McGregor, Chi-Lin Kuo, Thomas Beenakker, Chun-Sing Wong, Wendy A Offen, Zachary Armstrong, Bobby I Florea, Jeroen D Codee, Herman S. Overkleeft, Hans Aerts, Gideon Davies
      Exo--mannosidases are a broad class of stereochemically retaining hydrolases that are essential for the breakdown of complex carbohydrate substrates found in all kingdoms of life. Yet the detection of exo--mannosidases...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Rongalite-Induced Transition-Metal and Hydride-Free Reductive Aldol
           Reaction: A Rapid access to 3,3´- Disubstituted Oxindoles and Its
           Mechanistic Studies

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02284A, PaperSivaparwathi Golla, Naveenkumar Anugu, Swathi Jalagam, Hari Prasad Kokatla
      A transition-metal and hydride-free reductive aldol reaction has been developed for the synthesis of biologically active 3,3´-disubstituted oxindoles from isatin-derivatives using rongalite. In this protocol, rongalite plays the dual role...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Pd-Catalyzed Direct C−H Arylation of Pyrrolo[1,2-a]quinoxalines

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02248B, PaperDi Hao, Zhen Yang, Yali Liu, Yang Li, Chuntian Li, Yanlong Gu, Luigi Vaccaro, Jichang Liu, Ping Liu
      An efficient Pd-catalyzed direct C−H arylation of pyrrolo[1,2-a]quinoxalines with aryl iodides has been described, offering a selective route toward a series of 1-arylated and 1,3-diarylated pyrrolo[1,2-a]quinoxalines with good yields. This...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Alkynedicobalt Mediated Vinylogous Nazarov Reactions

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02256C, CommunicationSomaiah Almubayedh, James Green
      The SnCl4 mediated reactions of cross conjugated aryl enynone-Co2(CO)6 and dienynone-Co2(CO)6 complexes afford benzocycloheptynone complexes or cycloheptenynone complexes in a thermal vinylogous Nazarov process. The rate of ring closure is...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Asymmetric Synthesis of Isoxazole and Trifluoromethyl‐Containing
           3,2’‐Pyrrolidinyl Dispirooxindoles via Squaramide‐Catalysed [3 + 2]
           Cycloaddition Reactions

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02350K, PaperTong-Hao Li, Da-Ming Du
      A highly efficient squaramide‐catalysed asymmetric domino Michael/Mannich [3 + 2] cycloaddition of 3‐methyl‐4‐nitro‐5‐ isatylidenyl‐isoxazoles and N‐2,2,2‐trifluoroethylisatin ketimines was developed. A new class of complex and skeletondiversified isoxazole and trifluoromethyl‐containing 3,2’‐pyrrolidinyl...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Synthesis of 2-hydroxytetrahydrofurans by Wacker-type oxidation of
           1,1-disubstituted alkenes

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02277F, CommunicationRina Tanaka, Saki Komori, Yuhei Shimizu, Yasutaka Kataoka, Yasuyuki Ura
      1,1-Disubstituted alkenes feature high steric hindrance, which renders their Wacker-type oxidation difficult. We demonstrated the stereoselective synthesis of 2-hydroxytetrahydrofurans via the Wacker-type oxidation of 3-methyl-3-buten-1-ols by using a PdCl2(MeCN)2/NO/BQ catalyst...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Acylative kinetic resolution of racemic methyl-substituted cyclic
           alkylamines with 2,5-dioxopyrrolidin-1-yl (R)-2-phenoxypropanoate

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02099D, PaperDmitry Gruzdev, Sergey Vakarov, Marina Korolyova, Ekaterina V. Bartashevich, Andrey Tumashov, Evgeny Chulakov, Marina Ezhikova, Mikhail Kodess, Galina Levit, Victor Krasnov
      Diastereoselective acylation of a number of racemic methyl-substituted cyclic alkylamines with active esters of 2-phenoxypropanoic acid was studied in detail. Ester of (R)-2-phenoxypropanoic acid and N-hydroxysuccinimide was found to be...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • One-Step Synthesis of Indolizino[3,4,5-ab]isoindoles by
           Manganese(I)-Catalyzed C–H Activation: Structural Studies and
           Photophysical Properties

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02246F, CommunicationSara Cembellin, Ivan Maisuls, Constantin Gabriel Daniliuc, Helena Osthues, Nikos Doltsinis, Cristian Strassert, Frank Glorius
      Herein, a regioselective synthesis of indolizino[3,4,5-ab]isoindoles (INIs), a valuable class of heterocycles with interesting luminescence properties, is described using manganese(I)-catalyzed C−H activation. The reported transformation proceeds in a one-step procedure...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Microwave-assisted Palladium catalysed C-H acylation with aldehydes.
           Synthesis and diversification of 3-acylthiophenes

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02176A, PaperCarlos Santiago, Xabier Jimenez-Aberasturi, Eztizen Leicea, Marta G. Lete, Nuria Sotomayor, Esther Lete
      The use of MW allows the efficient palladium(II)-catalysed C-3 acylation of thiophenes with aldehydes via C(sp2)-H activation for the synthesis of (cyclo)alkyl/aryl thienyl ketones (43 examples). Compared to standard thermal...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Tandem Aza-Michael Addition―Vinylogous Aldol Condensation: Synthesis of
           N-Bridged Pyridine Fused Quinolones

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02087K, CommunicationLalitha Gummidi, Altaf Muddassar, Gangavaram VM Sharma, Murugesh V, Surisetti Suresh
      Herein, we present a tandem aza-Michael addition―vinylogous aldol condensation strategy for the synthesis of N-bridged pyridine fused quinolone derivatives from quinolones and ynones. The presented tandem transformation features the construction...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Enantioselective catalytic Povarov reactions

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02270A, Review ArticleJosé Clerigué, María Teresa Ramos, J. Carlos Menéndez
      Catalytic asymmetric Povarov protocols have undergone an explosive growth, especially in the last ten years, since the first example was published in 1996. The use of chiral Lewis and Brønsted...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Isoindolinone synthesis through Rh/Cu-catalyzed oxidative C-H/N-H
           annulation of N-methoxy benzamides with saturated ketones

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02166D, CommunicationXiao Du, Yuntao Hu, Darun Yang, Decai Huang, Wendi Yang, Hailong Wu, Huaiqing Zhao
      The synthesis of isoindolinones from N-methoxy benzamides and saturated ketones via a bimetallic tandem catalytic annulation has been accomplished. The reaction is catalyzed by a Rh/Cu-cocatalytic system and proceeds via...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Oxidative [4+2] Annulation of 1-Naphthols with Alkynes Accelerated by an
           Electron-Deficient Rhodium(III) Catalysts

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02181H, CommunicationAntônio Junio Araujo Dias, Hiroto Takahashi, Juntaro Nogami, Yuki Nagashima, Ken Tanaka
      The 1,3-diethoxycarbonyl-2,4,5-trimethylcyclopentadienyl (CpE) rhodium(III) complex displayed high efficacy in the catalytic oxidative annulation of 1-naphthols with internal alkynes under mild conditions. DFT calculations revealed that lower activation energies for the...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Effect of a cis-4-Aminopiperidine-3-carboxylic Acid (cis-APiC) Residue on
           Mixed-helical Folding of Unnatural Peptides

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02223G, PaperSunglim Choi, Jihyun Shim, Philjae Kang, Soo Hyuk Choi
      The α/β-peptide 11/9-helix and the β-peptide 12/10-helix belong to “mixed” helices, in which two types of hydrogen bonds with opposite directionality alternate along the helical axis. cis-2-Aminocyclohaxanecarboxylic acid (cis-ACHC) is...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Metal-Free Tandem Dehydrogenative α-Arylation Reaction of Propargylic
           Alcohols with 2-Alkynylbenzaldoximes toward the Synthesis of
           α-(4-Bromo-isoquinolin-1-yl)-propenone Skeletons

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02114A, CommunicationKhalil Alatat, Alireza Abbasi Kejani, Ali - Nikbakht, Hamid Reza Bijanzadeh, Saeed Balalaie
      A tandem reaction of 2-alkynylbenzaldoximes with propargylic alcohols has been developed for the synthesis of α-(4-bromo-isoquinolin-1-yl)-propenones. Employing 2-alkynylbenzaldoximes as a precursor in the presence of Br2 generates 4-Bromo-isoquinoline-N-oxides. Subsequently, dehydroxylation...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Metal-Free Sulfonylation of Arenes with N-Fluorobenzenesulfonimide via
           Cleavage of S-N Bonds: Expeditious Synthesis of Diarylsulfones

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02209A, CommunicationXiaohui Zhang, Yueji Feng, Yanyan Tuo, Qing-Zhong Zheng
      A novel metal-free sulfonylation of arenes with N-fluorobenzenesulfonimide (NFSI) toward the synthesis of diarylsulfones has been developed. The reaction represents a rare example of sulfonylation reaction using NFSI as efficient...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Rediscovering the Bacon’s Hydrazine/Phenylhydrazine Mediated Cyclization
           of 2,2’-Dicarbonylbi(hetero)aryls: Construction of
           (5-Azo)-/Indazolo[2,3-a]quinolines

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02207E, PaperPawan Surendra Dhote, Chepuri Ramana
      The hydrazine/phenylhydrazine mediated reductive dicarbonyl coupling reactions have been carried out under mild condition to arrive the construction of polycyclic aromatic compounds and azo-substituted polyaromatic compounds having a broad substrate...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • GlyConnect-Ugi: site-selective, multi-component glycoprotein conjugations
           through GlycoDelete expressed glycans

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Advance Article

      DOI : 10.1039/D1OB02299G, PaperKarel Thooft, Wander Van Breedam, Francis Santens, Elise Wyseure, Sandrine Vanmarcke, Simon Devos, Nico Callewaert, Annemieke Madder
      GlycoDelete proteins can be conveniently and site-selectively labeled upon oxidation of their unique glycan structure and their subsequent participation as aldehyde partner in a versatile multicomponent Ugi reaction.
      To cite this article before page numbers are assigned, use the
      DOI form of citation above.
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Time-economical synthesis of selenofunctionalized heterocycles via
           I2O5-mediated selenylative heterocyclization

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Advance Article

      DOI : 10.1039/D1OB02196F, PaperChen-Fan Zhou, Yun-Qian Zhang, Yong Ling, Liang Ming, Xia Xi, Gong-Qing Liu, Yanan Zhang
      A time-economical and robust synthesis of selenofunctionalized heterocycles by an I2O5-promoted selenylative heterocyclization of olefins with easily accessible diselenides is reported herein.
      To cite this article before page numbers are assigned, use the
      DOI form of citation above.
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Thioether-Directed Rh(III)-Catalyzed Peri-Selective Acyloxylation of
           Arenes

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02236A, CommunicationShang-Shi Zhang, Hui Xie, Song Jia-Lin, Chun-Yong Jiang, Yan-Xia Huang, Jun-Yi Zeng, Xu-Ge Liu, Fan Yang
      A thioether directed acyloxylation of arenes has been realized via Cp*Rh(III)-catalyzed C-H activation and subsequent coupling with carboxylic acids. This new method showed high functional group compatibility and broad substrate...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • 1,6-Addition of 1,2,3-NH triazoles to para-quinone methides: Facile access
           to highly selective N1 and N2 substituted triazoles

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Advance Article

      DOI : 10.1039/D1OB01717A, CommunicationVishakha Rai, Kavyashree P., Sarvesh S. Harmalkar, Sundar N. Dhuri, Mahagundappa R. Maddani
      Regioselective syntheses of N1 and N2 substituted triazoles via 1,6-addition of 1,2,3-NH triazole with p-QM were developed under mild reaction conditions. Isomerization of N1 to N2 substituted triazoles was also achieved in the presence of AlCl3.
      To cite this article before page numbers are assigned, use the
      DOI form of citation above.
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Synthesis of methylene-bridged α,β-unsaturated ketones: α-Csp3–H
           methylenation of aromatic ketones using Selectfluor as a mild oxidant

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Advance Article

      DOI : 10.1039/D1OB02043A, PaperYuan Zhang, Zhiqi Liu, Tingyu Zhu, Ying Huang, Weibin Fan, Deguang Huang
      A three starting material four component reaction is developed for the synthesis of α,β-unsaturated ketones and β-amino ketones. TMEDA is used a dual synthon to provide two carbons in the Selectfluor system.
      To cite this article before page numbers are assigned, use the
      DOI form of citation above.
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Four- and two-armed hetero porphyrin dimers: their specific recognition
           and self-sorting behaviours

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Advance Article

      DOI : 10.1039/D1OB01694F, PaperMasahiro Ueda, Masaki Kimura, Shinobu Miyagawa, Masaya Naito, Hikaru Takaya, Yuji Tokunaga
      Self-assembled/self-sorted hetero dimer capsules consisting of pairs of two- and four-armed porphyrins were constructed. Small and large aromatic guests were selectively recognized by two- and four-armed dimers, respectively.
      To cite this article before page numbers are assigned, use the
      DOI form of citation above.
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • A Unified Total Synthesis of Benzo[d][1,3]dioxole-type Benzylisoquinoline
           Alkaloids of Aporphines, Coptisines, and Dibenzopyrrocolines

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02258J, PaperJie Lv, Zhi-Hong Li, An-Jun Deng, Hai-Lin Qin
      The first total synthesis of (S)-(+)-ovigerine, (S)-(+)-N-formylovigerine, and (6aS,6a'S)-(+)-ovigeridimerine of aporphine alkaloids with benzo[d][1,3]dioxole structure feature was established. The strategy was based upon the well known Pd-catalyzed arylation to set...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Synthesis of aryl-heteroaryl derivatives via RhIII-catalyzed
           heteroarylation of arenes and heteroaromatic boronates

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02201F, PaperHuaiwei Wang, Jia-Xue Wu, DaCheng Li, Yu-Han Qiao, Qing-Xia Yao, Wen-Chan Sun, Jian-Min Dou
      An efficient RhIII-catalyzed strategy to construct aryl-heteroaryl derivatives via direct C−H heteroarylation of arenes and heteroaromatic boronates with removable ketoxime ether auxiliary has been disclosed. This protocol could tolerate various...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • An investigation of palladium-catalyzed Stille-type cross-coupling of
           nitroarenes in perylenediimide series

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02291A, CommunicationAline MAKHLOUTAH, Danylo Hatych, Thomas CHARTIER, Lou ROCARD, Antoine Goujon, François-Xavier Felpin, pietrick hudhomme
      We report herein an unprecedented palladium-catalyzed cross-coupling reaction between mononitro-perylenediimide (PDI) and various arylstannanes. Optimized conditions developed with this Stille-type reaction allow the grafting of (hetero)aryls of various electronic nature...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Cu(OAc)2/DABCO-mediated domino reaction of vinyl malononitriles with
           cyclic sulfamidate imines: access to 6-hydroxyaryl-2-aminonicotinonitriles
           

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02095A, CommunicationS Banuprakash Goud, Soumitra Guin, Meher Prakash, Sampak Samanta
      A novel Cu(II)-salt/DABCO-mediated one-pot access to a myriad of highly-substituted biologically relevant 2-aminonicotinonitriles possessing a resourceful phenolic moiety with satisfactory yields is reported. This method involves cyclic sulfamidate imines as...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Rhodium(III)-catalyzed oxidative annulation of isoquinolones with allyl
           alcohols: synthesis of isoindolo[2,1-b]isoquinolin-5(7H)-ones

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02305E, CommunicationJinyuan Jiang, Jidan Liu, Zhenke Yang, Jieying Zheng, Xin Tian, Liyao Zheng, Zhao-Qing Liu
      An efficient rhodium(III)-catalyzed direct C-H oxidative annulation of isoquinolones with allyl alcohols as C1 synthons has been successfully developed. This protocol enables the straightforward synthesis of structurally diverse isoindolo[2,1-b]isoquinolin-5(7H)-ones with...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Palladium-Catalyzed anti-Markovnikov Oxidative Acetalization of Activated
           Olefins with Iron(III) Sulphate as Benign Reoxidant

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02227J, PaperRodney Agustinho Fernandes, Sandhya Singh Yadav, Praveen Kumar
      This paper discloses the efficient palladium-catalyzed anti-Markovnikov oxidative acetalization of activated terminal olefins with iron(III) sulfate as benign reoxidant. This methodology depicts mild reaction conditions, high regioselectivity toward anti-Makovnikov products...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Reactivity Switch-Over of 4-Hydroxydithiocoumarin Under Various Conditions
           and Their Application in Organic Synthesis

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB01357B, Review ArticleMd. Belal, Santa Mondal, Sabina Yashmin, Abu Taleb Khan
      4-hydroxydithiocoumarin is a valuable organic precursor to architect important heterocycles. The three different reactive nucleophilic sites at the 4-hydroxydithiocoumarins display intriguing regioselectivity in its reaction towards various electro-philes. Previously, 4-hydroxydithiocoumarins...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
  • Synthesis of Rhein and Diacerein: A Chemoenzymatic Approach using Anthrol
           Reductase of Talaromyces islandicus

    • Free pre-print version: Loading...

      Abstract: Org. Biomol. Chem., 2022, Accepted Manuscript

      DOI : 10.1039/D1OB02202D, CommunicationAnshul Rajput, Amit Mondal, Satyendra Kumar Pandey, Syed Masood Husain
      Herein, we report two methods for the synthesis of osteoarthritis drug, rhein and its prodrug diacerein using a chemoenzymatic approach. The strategy relies on the use of an NADPH-dependent anthrol...
      The content of this RSS Feed (c) The Royal Society of Chemistry
       
 
JournalTOCs
School of Mathematical and Computer Sciences
Heriot-Watt University
Edinburgh, EH14 4AS, UK
Email: journaltocs@hw.ac.uk
Tel: +00 44 (0)131 4513762
 


Your IP address: 52.23.215.230
 
Home (Search)
API
About JournalTOCs
News (blog, publications)
JournalTOCs on Twitter   JournalTOCs on Facebook

JournalTOCs © 2009-